Last reviewed · How we verify

penile nerve block with bupivacaine

University of Colorado, Denver · FDA-approved active Small molecule

Bupivacaine blocks sodium channels in nerve fibers to provide local anesthesia and pain relief in the penile region.

Bupivacaine blocks sodium channels in nerve fibers to provide local anesthesia and pain relief in the penile region. Used for Local anesthesia for penile surgical procedures and interventions.

At a glance

Generic namepenile nerve block with bupivacaine
SponsorUniversity of Colorado, Denver
Drug classLocal anesthetic
TargetVoltage-gated sodium channels
ModalitySmall molecule
Therapeutic areaAnesthesia / Urology
PhaseFDA-approved

Mechanism of action

Bupivacaine is a local anesthetic that reversibly inhibits sodium influx into nerve cells, preventing depolarization and blocking nerve conduction. When administered as a penile nerve block, it anesthetizes the dorsal nerves of the penis and surrounding sensory nerves, providing localized pain relief without systemic effects. This allows for pain-free surgical or procedural intervention on penile tissue.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results