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OROS MPH

Ortho-McNeil Janssen Scientific Affairs, LLC · FDA-approved active Small molecule

OROS MPH is an extended-release formulation of methylphenidate that provides sustained dopamine and norepinephrine reuptake inhibition throughout the day.

OROS MPH is an extended-release formulation of methylphenidate that provides sustained dopamine and norepinephrine reuptake inhibition throughout the day. Used for Attention-deficit/hyperactivity disorder (ADHD) in children and adults.

At a glance

Generic nameOROS MPH
Also known asConcerta
SponsorOrtho-McNeil Janssen Scientific Affairs, LLC
Drug classCentral nervous system stimulant; dopamine-norepinephrine reuptake inhibitor
TargetDopamine transporter (DAT); norepinephrine transporter (NET)
ModalitySmall molecule
Therapeutic areaPsychiatry / Neurology
PhaseFDA-approved

Mechanism of action

Methylphenidate is a central nervous system stimulant that blocks the reuptake of dopamine and norepinephrine at the presynaptic neuron, increasing their availability in the synaptic cleft. The OROS (osmotic release oral system) technology delivers the drug in a controlled, extended manner over approximately 12 hours, providing consistent therapeutic levels and reducing the need for multiple daily doses. This mechanism enhances attention, focus, and impulse control in patients with attention-deficit/hyperactivity disorder.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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