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Opdivo (nivolumab)
Opdivo works by blocking the PD-1 receptor on immune cells, allowing them to attack cancer cells.
Opdivo (nivolumab) is a programmed death receptor-1 blocking antibody developed by Bristol Myers Squibb. It targets the programmed cell death protein 1 (PD-1) to inhibit cancer cell growth. Opdivo is approved for various cancer indications, including melanoma, Hodgkin lymphoma, and renal cell carcinoma. The drug has a half-life of 25 days and is patented by Bristol Myers Squibb. Key safety considerations include immune-mediated adverse reactions and infusion-related reactions.
At a glance
| Generic name | nivolumab |
|---|---|
| Sponsor | Bristol-Myers Squibb |
| Drug class | Programmed Death Receptor-1 Blocking Antibody [EPC] |
| Target | Programmed cell death protein 1 |
| Modality | Monoclonal antibody |
| Therapeutic area | Oncology |
| Phase | FDA-approved |
| First approval | 2014 |
| Annual revenue | 9200 |
Mechanism of action
Binding of the PD-1 ligands, PD-L1 and PD-L2, to the PD-1 receptor found on cells, inhibits T-cell proliferation and cytokine production. Upregulation of PD-1 ligands occurs in some tumors and signaling through this pathway can contribute to inhibition of active T-cell immune surveillance of tumors. Nivolumab is human immunoglobulin G4 (IgG4) monoclonal antibody that binds to the PD-1 receptor and blocks its interaction with PD-L1 and PD-L2, releasing PD-1 pathway-mediated inhibition of the immune response, including the anti-tumor immune response. In syngeneic mouse tumor models, blocking PD-1 activity resulted in decreased tumor growth.Combined nivolumab (anti-PD-1) and ipilimumab (anti-CTLA-4) mediated inhibition results in enhanced T-cell function that is greater than the effects of either antibody alone, and results in improved anti-tumor responses in metastatic melanoma and advanced RCC. In murine syngeneic tumor models, dual blockade of PD-1 and CTLA-4
Approved indications
- Advanced melanoma with tumour cell PD-L1 expression below 1%
- Classical Hodgkin lymphoma
- Head and neck cancer
- Malignant tumor of esophagus
- Malignant tumor of stomach
- Metastatic malignant melanoma
- Metastatic renal cell carcinoma
- Microsatellite instability-high colorectal cancer
- Non-small cell lung cancer
- Postoperative adjuvant therapy for urothelial carcinoma
- Squamous cell carcinoma of lung
- Transitional cell carcinoma
- Unresectable advanced or recurrent malignant pleural mesothelioma
- Unresectable, advanced or recurrent gastric cancer
Common side effects
- Fatigue
- Rash
- Musculoskeletal pain
- Pruritus
- Diarrhea
- Nausea
- Asthenia
- Cough
- Dyspnea
- Constipation
- Decreased appetite
- Back pain
Key clinical trials
- An Investigational Immuno-therapy Trial of Nivolumab, or Nivolumab Plus Ipilimumab, or Nivolumab Plus Platinum-doublet Chemotherapy, Compared to Platinum Doublet Chemotherapy in Patients With Stage IV Non-Small Cell Lung Cancer (NSCLC) (PHASE3)
- Study of Nivolumab Combined With Ipilimumab Versus Pemetrexed and Cisplatin or Carboplatin as First Line Therapy in Unresectable Pleural Mesothelioma Patients (PHASE3)
- A Study of Nivolumab and Ipilimumab Combined With Chemotherapy Compared to Chemotherapy Alone in First Line NSCLC (PHASE3)
- Study of Nivolumab (BMS-936558) Compared With Dacarbazine in Untreated, Unresectable, or Metastatic Melanoma (PHASE3)
- Efficacy Study of Nivolumab Compared to Ipilimumab in Prevention of Recurrence of Melanoma After Complete Resection of Stage IIIb/c or Stage IV Melanoma (PHASE3)
- Nivolumab Combined With Ipilimumab Versus Sunitinib in Previously Untreated Advanced or Metastatic Renal Cell Carcinoma (CheckMate 214) (PHASE3)
- A Study to Compare BMS-936558 to the Physician's Choice of Either Dacarbazine or Carboplatin and Paclitaxel in Advanced Melanoma Patients That Have Progressed Following Anti-CTLA-4 Therapy (CheckMate 037) (PHASE3)
- Phase 3 Study of Nivolumab or Nivolumab Plus Ipilimumab Versus Ipilimumab Alone in Previously Untreated Advanced Melanoma (CheckMate 067) (PHASE3)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| FDA label | Mechanism, indications, dosing, boxed warnings, drug interactions |
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
| SEC EDGAR | Revenue + earnings |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Opdivo CI brief — competitive landscape report
- Opdivo updates RSS · CI watch RSS
- Bristol-Myers Squibb portfolio CI