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Midazolam sedation

University of Liege · FDA-approved active Small molecule

Midazolam sedation is a Benzodiazepine Small molecule drug developed by University of Liege. It is currently FDA-approved for Procedural sedation and anxiolysis, Induction of general anesthesia, Acute anxiety and agitation.

Midazolam is a benzodiazepine that enhances the inhibitory effects of GABA at GABA-A receptors in the central nervous system, producing sedation and anxiolysis.

Midazolam is a benzodiazepine that enhances the inhibitory effects of GABA at GABA-A receptors in the central nervous system, producing sedation and anxiolysis. Used for Procedural sedation and anxiolysis, Induction of general anesthesia, Acute agitation and anxiety management.

At a glance

Generic nameMidazolam sedation
SponsorUniversity of Liege
Drug classBenzodiazepine
TargetGABA-A receptor
ModalitySmall molecule
Therapeutic areaAnesthesia/Sedation
PhaseFDA-approved

Mechanism of action

Midazolam binds to GABA-A receptors and potentiates the effect of the inhibitory neurotransmitter GABA, leading to increased chloride ion influx and neuronal hyperpolarization. This results in depression of the central nervous system, manifesting as sedation, anxiolysis, muscle relaxation, and anticonvulsant effects. The drug is commonly used for procedural sedation and anesthesia induction due to its rapid onset and short duration of action.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Midazolam sedation

What is Midazolam sedation?

Midazolam sedation is a Benzodiazepine drug developed by University of Liege, indicated for Procedural sedation and anxiolysis, Induction of general anesthesia, Acute anxiety and agitation.

How does Midazolam sedation work?

Midazolam is a benzodiazepine that enhances the inhibitory effects of GABA at GABA-A receptors in the central nervous system, producing sedation and anxiolysis.

What is Midazolam sedation used for?

Midazolam sedation is indicated for Procedural sedation and anxiolysis, Induction of general anesthesia, Acute anxiety and agitation, Seizure management.

Who makes Midazolam sedation?

Midazolam sedation is developed and marketed by University of Liege (see full University of Liege pipeline at /company/university-of-liege).

What drug class is Midazolam sedation in?

Midazolam sedation belongs to the Benzodiazepine class. See all Benzodiazepine drugs at /class/benzodiazepine.

What development phase is Midazolam sedation in?

Midazolam sedation is FDA-approved (marketed).

What are the side effects of Midazolam sedation?

Common side effects of Midazolam sedation include Respiratory depression, Hypotension, Oversedation, Amnesia, Paradoxical reaction (agitation, disinhibition), Headache.

What does Midazolam sedation target?

Midazolam sedation targets GABA-A receptor and is a Benzodiazepine.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing