Last reviewed · How we verify
midazolam in children premedication
midazolam in children premedication is a Benzodiazepine Small molecule drug developed by Azienda Ospedaliera Universitaria Policlinico "G. Martino". It is currently FDA-approved for Premedication and anxiolysis in children undergoing surgical or diagnostic procedures, Sedation in pediatric patients.
Midazolam is a benzodiazepine that enhances inhibitory GABAergic neurotransmission in the central nervous system to produce sedation and anxiolysis.
Midazolam is a benzodiazepine that enhances inhibitory GABAergic neurotransmission in the central nervous system to produce sedation and anxiolysis. Used for Premedication and anxiolysis in children undergoing surgical or diagnostic procedures, Sedation in pediatric patients.
At a glance
| Generic name | midazolam in children premedication |
|---|---|
| Sponsor | Azienda Ospedaliera Universitaria Policlinico "G. Martino" |
| Drug class | Benzodiazepine |
| Target | GABA-A receptor |
| Modality | Small molecule |
| Therapeutic area | Anesthesia/Sedation |
| Phase | FDA-approved |
Mechanism of action
Midazolam binds to benzodiazepine receptors on GABA-A receptors, increasing the frequency of chloride channel opening and hyperpolarizing neuronal membranes. This results in reduced neuronal excitability and produces sedative, anxiolytic, and amnestic effects. In pediatric premedication, it reduces anxiety and facilitates smoother induction of anesthesia.
Approved indications
- Premedication and anxiolysis in children undergoing surgical or diagnostic procedures
- Sedation in pediatric patients
Common side effects
- Respiratory depression
- Hypotension
- Paradoxical agitation
- Oversedation
- Emergence delirium
Key clinical trials
- Comparison of Oral Dexmedetomidine, Ketamine Versus Midazolam for Premedication in Children Undergoing Injuinal Surgeries (NA)
- Melatonin vs Midazolam in Children Undergoing Tonsillectomy (PHASE3)
- Assessment of Endotracheal Tube Temperature Effects in Children Undergoing Adenotonsillectomy (NA)
- Intranasal Dexmedetomidine Versus Oral Midazolam Premedication for Postoperative Negative Behavior Changes in Children (PHASE4)
- Intranasal Dexmedetomidine, Ketamine or Midazolam for Anxiety and Respiratory Complications in Children (NA)
- Use Of Midazolam In Premedication Of Pediatric Patients (NA)
- Comparing Two Doses of Midazolam With Added Dexmedetomidine for Kids Before Surgery (PHASE2)
- Using of Virtual Reality to Relieve Procedural Pain in Pediatric Oncology. (NA)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- midazolam in children premedication CI brief — competitive landscape report
- midazolam in children premedication updates RSS · CI watch RSS
- Azienda Ospedaliera Universitaria Policlinico "G. Martino" portfolio CI
Frequently asked questions about midazolam in children premedication
What is midazolam in children premedication?
How does midazolam in children premedication work?
What is midazolam in children premedication used for?
Who makes midazolam in children premedication?
What drug class is midazolam in children premedication in?
What development phase is midazolam in children premedication in?
What are the side effects of midazolam in children premedication?
What does midazolam in children premedication target?
Related
- Drug class: All Benzodiazepine drugs
- Target: All drugs targeting GABA-A receptor
- Manufacturer: Azienda Ospedaliera Universitaria Policlinico "G. Martino" — full pipeline
- Therapeutic area: All drugs in Anesthesia/Sedation
- Indication: Drugs for Premedication and anxiolysis in children undergoing surgical or diagnostic procedures
- Indication: Drugs for Sedation in pediatric patients
- Compare: midazolam in children premedication vs similar drugs
- Pricing: midazolam in children premedication cost, discount & access