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low dose peroral misoprostol

University Medical Centre Ljubljana · FDA-approved active Small molecule

Misoprostol is a prostaglandin E1 analogue that stimulates gastric mucus secretion and reduces gastric acid production to protect the gastrointestinal mucosa.

Misoprostol is a prostaglandin E1 analogue that stimulates gastric mucus secretion and reduces gastric acid production to protect the gastrointestinal mucosa. Used for Prevention of NSAID-induced gastric ulcers, Gastroprotection in patients requiring chronic NSAID therapy.

At a glance

Generic namelow dose peroral misoprostol
SponsorUniversity Medical Centre Ljubljana
Drug classProstaglandin E1 analogue
TargetProstaglandin E receptor (EP receptor)
ModalitySmall molecule
Therapeutic areaGastroenterology
PhaseFDA-approved

Mechanism of action

Misoprostol binds to prostaglandin receptors on gastric epithelial cells, enhancing mucus and bicarbonate secretion while simultaneously decreasing gastric acid secretion. At low oral doses, it is used primarily for gastroprotection, particularly in patients taking nonsteroidal anti-inflammatory drugs (NSAIDs) who are at risk for peptic ulcer disease. The drug also has uterotonic properties at higher doses, but low-dose formulations are marketed for GI protection.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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