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Lisinopril + HCTZ

St. Paul Heart Clinic · Phase 3 active Small molecule

Lisinopril inhibits angiotensin-converting enzyme to reduce blood pressure, while HCTZ is a thiazide diuretic that lowers blood pressure by reducing fluid volume and sodium reabsorption.

Lisinopril inhibits angiotensin-converting enzyme to reduce blood pressure, while HCTZ is a thiazide diuretic that lowers blood pressure by reducing fluid volume and sodium reabsorption. Used for Hypertension, Heart failure with reduced ejection fraction.

At a glance

Generic nameLisinopril + HCTZ
Also known asPrinivil, Hydrochlorothiazide
SponsorSt. Paul Heart Clinic
Drug classACE inhibitor + thiazide diuretic combination
TargetAngiotensin-converting enzyme (ACE); sodium-chloride cotransporter (NCCT)
ModalitySmall molecule
Therapeutic areaCardiovascular
PhasePhase 3

Mechanism of action

Lisinopril blocks ACE, preventing conversion of angiotensin I to angiotensin II, thereby reducing vasoconstriction and aldosterone secretion. HCTZ acts as a thiazide diuretic, increasing urinary sodium and water excretion to decrease blood volume and peripheral vascular resistance. Together, these complementary mechanisms provide synergistic antihypertensive effects.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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