Last reviewed · How we verify

lidocaine+systemic tramadol

Bagcilar Training and Research Hospital · Phase 3 active Small molecule

Lidocaine is a local anesthetic that blocks nerve signals, while tramadol is a weak opioid agonist and norepinephrine reuptake inhibitor that relieves pain.

Lidocaine is a local anesthetic that blocks nerve signals, while tramadol is a weak opioid agonist and norepinephrine reuptake inhibitor that relieves pain. Used for Moderate to severe pain, Postoperative pain.

At a glance

Generic namelidocaine+systemic tramadol
Also known astramadol
SponsorBagcilar Training and Research Hospital
Drug classLocal anesthetic and weak opioid agonist
TargetMu-opioid receptor, Norepinephrine transporter
ModalitySmall molecule
Therapeutic areaPain management
PhasePhase 3

Mechanism of action

Lidocaine works by stabilizing the neuronal membrane and blocking the generation and conduction of nerve impulses. Tramadol, on the other hand, binds to mu-opioid receptors and inhibits the reuptake of norepinephrine, resulting in analgesia.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results