Last reviewed · How we verify

L-Histidine

University of Miami · FDA-approved active Small molecule

L-Histidine is an essential amino acid that serves as a precursor for histamine and other bioactive compounds involved in immune regulation, gastric acid secretion, and vasodilation.

L-Histidine is an essential amino acid that serves as a precursor for histamine and other bioactive compounds involved in immune regulation, gastric acid secretion, and vasodilation. Used for Histidine deficiency or supplementation in medical nutrition, Potential adjunctive use in immune support or inflammatory conditions.

At a glance

Generic nameL-Histidine
Also known asHistamine
SponsorUniversity of Miami
Drug classAmino acid supplement
ModalitySmall molecule
Therapeutic areaNutritional/Metabolic
PhaseFDA-approved

Mechanism of action

L-Histidine is metabolized to histamine, which plays critical roles in immune responses, inflammation, gastric acid production, and vascular tone regulation. It also participates in protein synthesis and serves as a precursor for other important molecules including carnosine and anserine. As a nutritional supplement or pharmaceutical agent, L-Histidine may be used to support immune function, improve gastric health, or address histidine deficiency states.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

Competitive intelligence

For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape: