Last reviewed · How we verify

KK8398

Kyowa Kirin Co., Ltd. · Phase 3 active Small molecule

KK8398 is a complement C5a receptor antagonist that blocks the C5a-C5aR1 signaling pathway to reduce inflammatory cell recruitment and activation.

KK8398 is a complement C5a receptor antagonist that blocks the C5a-C5aR1 signaling pathway to reduce inflammatory cell recruitment and activation. Used for Autoimmune/inflammatory conditions (specific indication under investigation in phase 3).

At a glance

Generic nameKK8398
SponsorKyowa Kirin Co., Ltd.
Drug classComplement C5a receptor antagonist
TargetC5aR1 (C5a receptor 1)
ModalitySmall molecule
Therapeutic areaImmunology
PhasePhase 3

Mechanism of action

By antagonizing the C5a receptor (C5aR1), KK8398 inhibits complement-mediated inflammation, which plays a key role in various inflammatory and autoimmune diseases. This mechanism reduces the chemotactic activity of C5a, thereby decreasing neutrophil and other immune cell infiltration into affected tissues and limiting downstream inflammatory cascades.

Approved indications

Common side effects

No common side effects on file.

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

Competitive intelligence

For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape: