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Keppra® extended release formulation - XR

UCB Pharma · Phase 3 active Small molecule

Levetiracetam binds to synaptic vesicle protein 2A (SV2A) to reduce neuronal excitability and prevent seizure propagation.

Levetiracetam binds to synaptic vesicle protein 2A (SV2A) to reduce neuronal excitability and prevent seizure propagation. Used for Adjunctive therapy for partial-onset seizures, Adjunctive therapy for myoclonic seizures in patients with juvenile myoclonic epilepsy, Adjunctive therapy for primary generalized tonic-clonic seizures.

At a glance

Generic nameKeppra® extended release formulation - XR
Also known asLevetiracetam XR
SponsorUCB Pharma
Drug classAntiepileptic drug (AED)
TargetSV2A (synaptic vesicle protein 2A)
ModalitySmall molecule
Therapeutic areaNeurology
PhasePhase 3

Mechanism of action

Levetiracetam's exact mechanism is not fully elucidated, but it is believed to work primarily through binding to SV2A, a protein involved in synaptic vesicle exocytosis. This binding may modulate neurotransmitter release and reduce abnormal neuronal firing. Unlike many other antiepileptic drugs, it does not directly affect sodium or calcium channels or enhance GABA inhibition.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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