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Janumet, Lantus
Janumet combines sitagliptin (a DPP-4 inhibitor) with metformin to lower blood glucose by increasing incretin levels and reducing hepatic glucose production, while Lantus is a long-acting basal insulin that provides steady glucose control.
Janumet combines sitagliptin (a DPP-4 inhibitor) with metformin to lower blood glucose by increasing incretin levels and reducing hepatic glucose production, while Lantus is a long-acting basal insulin that provides steady glucose control. Used for Type 2 diabetes mellitus (Janumet as oral agent; Lantus as basal insulin therapy).
At a glance
| Generic name | Janumet, Lantus |
|---|---|
| Sponsor | Chinese University of Hong Kong |
| Drug class | DPP-4 inhibitor + biguanide (Janumet); long-acting basal insulin (Lantus) |
| Target | DPP-4 enzyme, metformin (AMPK pathway), insulin receptor (Lantus) |
| Modality | Small molecule |
| Therapeutic area | Diabetes |
| Phase | FDA-approved |
Mechanism of action
Janumet works through dual action: sitagliptin inhibits dipeptidyl peptidase-4 to prolong GLP-1 and GIP activity, stimulating insulin secretion in response to meals, while metformin decreases hepatic glucose output and improves insulin sensitivity. Lantus (insulin glargine) is a basal insulin analog that provides continuous glucose-lowering effect over 24 hours by mimicking the body's natural background insulin secretion. Together, these agents address multiple pathways in type 2 diabetes pathophysiology.
Approved indications
- Type 2 diabetes mellitus (Janumet as oral agent; Lantus as basal insulin therapy)
Common side effects
- Hypoglycemia
- Gastrointestinal disturbance (nausea, diarrhea)
- Upper respiratory tract infection
- Headache
- Injection site reactions (Lantus)
Key clinical trials
- Remission Evaluation of a Metabolic Intervention in Type 2 Diabetes With Sitagliptin (REMIT-Sita) (PHASE3)
- Metformin and Sitagliptin Therapy for Adult Patients With Type 2 Diabetes Admitted to the General Medical Unit (PHASE4)
- Randomized Sitagliptin Withdrawal Study (MK-0431-845) (PHASE3)
- Safety and Efficacy of Ertugliflozin in the Treatment of Participants With Type 2 Diabetes Mellitus Who Have Inadequate Glycemic Control on Metformin and Sitagliptin (MK-8835-006; VERTIS SITA2) (PHASE3)
- Sitagliptin Therapy in Hospitalized Patients With Type 2 Diabetes (PHASE4)
- JanUmet Before Insulin Lantus In Eastern Population Evaluation Program (JUBILEE) In Type 2 Diabetic Patients (PHASE4)
- ß-Cell Function and Glycemic Control in Newly Diagnosed Type 2 Diabetic Patients With Moderate Hyperglycemia (PHASE4)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Janumet, Lantus CI brief — competitive landscape report
- Janumet, Lantus updates RSS · CI watch RSS
- Chinese University of Hong Kong portfolio CI