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Intravenous amiodarone(2)

Instituto de Cardiología y Medicina Vascular Hospital Zambrano-Hellion Tec Salud · FDA-approved active Small molecule

Intravenous amiodarone(2) is a Class III antiarrhythmic agent Small molecule drug developed by Instituto de Cardiología y Medicina Vascular Hospital Zambrano-Hellion Tec Salud. It is currently FDA-approved for Atrial fibrillation with rapid ventricular response, Ventricular tachycardia, Ventricular fibrillation. Also known as: 72 hour amiodarone.

Intravenous amiodarone is a Class III antiarrhythmic agent that blocks potassium channels and prolongs the action potential duration and refractory period to restore normal heart rhythm.

Intravenous amiodarone is a Class III antiarrhythmic agent that blocks potassium channels and prolongs the action potential duration and refractory period to restore normal heart rhythm. Used for Atrial fibrillation with rapid ventricular response, Ventricular tachycardia, Ventricular fibrillation.

At a glance

Generic nameIntravenous amiodarone(2)
Also known as72 hour amiodarone
SponsorInstituto de Cardiología y Medicina Vascular Hospital Zambrano-Hellion Tec Salud
Drug classClass III antiarrhythmic agent
TargetPotassium channels (hERG), sodium channels, beta-adrenergic receptors, calcium channels
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved

Mechanism of action

Amiodarone works primarily through potassium channel blockade, which delays repolarization and extends the action potential duration. It also has properties of all four Vaughan-Williams antiarrhythmic classes, including sodium channel blockade, beta-adrenergic antagonism, and calcium channel inhibition. This multi-channel activity makes it effective for suppressing various cardiac arrhythmias.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Intravenous amiodarone(2)

What is Intravenous amiodarone(2)?

Intravenous amiodarone(2) is a Class III antiarrhythmic agent drug developed by Instituto de Cardiología y Medicina Vascular Hospital Zambrano-Hellion Tec Salud, indicated for Atrial fibrillation with rapid ventricular response, Ventricular tachycardia, Ventricular fibrillation.

How does Intravenous amiodarone(2) work?

Intravenous amiodarone is a Class III antiarrhythmic agent that blocks potassium channels and prolongs the action potential duration and refractory period to restore normal heart rhythm.

What is Intravenous amiodarone(2) used for?

Intravenous amiodarone(2) is indicated for Atrial fibrillation with rapid ventricular response, Ventricular tachycardia, Ventricular fibrillation, Supraventricular tachycardia.

Who makes Intravenous amiodarone(2)?

Intravenous amiodarone(2) is developed and marketed by Instituto de Cardiología y Medicina Vascular Hospital Zambrano-Hellion Tec Salud (see full Instituto de Cardiología y Medicina Vascular Hospital Zambrano-Hellion Tec Salud pipeline at /company/instituto-de-cardiolog-a-y-medicina-vascular-hospital-zambrano-hellion-tec-salud).

Is Intravenous amiodarone(2) also known as anything else?

Intravenous amiodarone(2) is also known as 72 hour amiodarone.

What drug class is Intravenous amiodarone(2) in?

Intravenous amiodarone(2) belongs to the Class III antiarrhythmic agent class. See all Class III antiarrhythmic agent drugs at /class/class-iii-antiarrhythmic-agent.

What development phase is Intravenous amiodarone(2) in?

Intravenous amiodarone(2) is FDA-approved (marketed).

What are the side effects of Intravenous amiodarone(2)?

Common side effects of Intravenous amiodarone(2) include Hypotension, Bradycardia, Phlebitis at injection site, Nausea, Pulmonary toxicity (chronic use), Thyroid dysfunction (chronic use).

What does Intravenous amiodarone(2) target?

Intravenous amiodarone(2) targets Potassium channels (hERG), sodium channels, beta-adrenergic receptors, calcium channels and is a Class III antiarrhythmic agent.

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