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Intrastromal voriconazole

University of California, San Francisco · Phase 3 active Small molecule

Intrastromal voriconazole is an antifungal agent delivered directly into the corneal stroma to treat fungal keratitis by inhibiting fungal cell wall synthesis.

Intrastromal voriconazole is an antifungal agent delivered directly into the corneal stroma to treat fungal keratitis by inhibiting fungal cell wall synthesis. Used for Fungal keratitis (corneal fungal infection).

At a glance

Generic nameIntrastromal voriconazole
SponsorUniversity of California, San Francisco
Drug classTriazole antifungal
TargetLanosterol 14α-demethylase (CYP51)
ModalitySmall molecule
Therapeutic areaOphthalmology / Infectious Disease
PhasePhase 3

Mechanism of action

Voriconazole is a triazole antifungal that inhibits lanosterol 14α-demethylase, a key enzyme in fungal ergosterol synthesis, disrupting the fungal cell membrane. When administered intrastromally (directly into corneal tissue), it achieves high local concentrations to treat corneal fungal infections that are difficult to penetrate with topical or systemic administration.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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