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Intraduodenal denatonium benzoate

Universitaire Ziekenhuizen KU Leuven · FDA-approved active Small molecule

Denatonium benzoate is a bitter-tasting compound administered intraduodenally that triggers taste receptors to elicit a protective reflex and modify gastrointestinal function.

Denatonium benzoate is a bitter-tasting compound administered intraduodenally that triggers taste receptors to elicit a protective reflex and modify gastrointestinal function. Used for Dumping syndrome (post-bariatric surgery or post-gastrectomy).

At a glance

Generic nameIntraduodenal denatonium benzoate
Also known asIG DB
SponsorUniversitaire Ziekenhuizen KU Leuven
Drug classBitter taste receptor agonist
TargetBitter taste receptors (T2Rs), particularly TAS2R family members
ModalitySmall molecule
Therapeutic areaGastroenterology
PhaseFDA-approved

Mechanism of action

Denatonium benzoate is one of the most bitter substances known and activates bitter taste receptors (T2Rs) in the duodenum when delivered directly into the small intestine. This activation triggers vagal afferent signaling and local enteric nervous system responses that modulate gastric emptying, intestinal motility, and potentially nutrient absorption. The bitter taste reflex is thought to provide a protective mechanism against ingestion of potentially toxic substances.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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