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imidafenacin, KRP-197/ONO-8025

Ono Pharmaceutical Co. Ltd · Phase 3 active Small molecule

imidafenacin, KRP-197/ONO-8025 is a Antimuscarinic Small molecule drug developed by Ono Pharmaceutical Co. Ltd. It is currently in Phase 3 development for Overactive bladder (urge urinary incontinence).

Imidafenacin is an antimuscarinic agent that acts as a selective M3 receptor antagonist.

Imidafenacin is an antimuscarinic agent that acts as a selective M3 receptor antagonist. Used for Overactive bladder (urge urinary incontinence).

At a glance

Generic nameimidafenacin, KRP-197/ONO-8025
SponsorOno Pharmaceutical Co. Ltd
Drug classAntimuscarinic
TargetM3 receptor
ModalitySmall molecule
Therapeutic areaUrology
PhasePhase 3

Mechanism of action

By blocking the M3 receptor, imidafenacin reduces bladder contractions and decreases the frequency of urge urinary incontinence episodes. This mechanism of action is specific to the M3 receptor subtype, which is primarily responsible for bladder contractions. As a result, imidafenacin provides targeted relief for patients with overactive bladder symptoms.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about imidafenacin, KRP-197/ONO-8025

What is imidafenacin, KRP-197/ONO-8025?

imidafenacin, KRP-197/ONO-8025 is a Antimuscarinic drug developed by Ono Pharmaceutical Co. Ltd, indicated for Overactive bladder (urge urinary incontinence).

How does imidafenacin, KRP-197/ONO-8025 work?

Imidafenacin is an antimuscarinic agent that acts as a selective M3 receptor antagonist.

What is imidafenacin, KRP-197/ONO-8025 used for?

imidafenacin, KRP-197/ONO-8025 is indicated for Overactive bladder (urge urinary incontinence).

Who makes imidafenacin, KRP-197/ONO-8025?

imidafenacin, KRP-197/ONO-8025 is developed by Ono Pharmaceutical Co. Ltd (see full Ono Pharmaceutical Co. Ltd pipeline at /company/ono-pharmaceutical-co-ltd).

What drug class is imidafenacin, KRP-197/ONO-8025 in?

imidafenacin, KRP-197/ONO-8025 belongs to the Antimuscarinic class. See all Antimuscarinic drugs at /class/antimuscarinic.

What development phase is imidafenacin, KRP-197/ONO-8025 in?

imidafenacin, KRP-197/ONO-8025 is in Phase 3.

What are the side effects of imidafenacin, KRP-197/ONO-8025?

Common side effects of imidafenacin, KRP-197/ONO-8025 include Dry mouth, Constipation, Headache.

What does imidafenacin, KRP-197/ONO-8025 target?

imidafenacin, KRP-197/ONO-8025 targets M3 receptor and is a Antimuscarinic.

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