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GEMIGLIPTIN LS15-0444

Sanofi · Phase 3 active Small molecule

Gemigliptin is a dipeptidyl peptidase-4 (DPP-4) inhibitor that increases levels of incretin hormones to stimulate insulin secretion in response to glucose.

Gemigliptin is a dipeptidyl peptidase-4 (DPP-4) inhibitor that increases levels of incretin hormones to stimulate insulin secretion in response to glucose. Used for Type 2 diabetes mellitus.

At a glance

Generic nameGEMIGLIPTIN LS15-0444
Also known asZemiglo
SponsorSanofi
Drug classDPP-4 inhibitor
TargetDPP-4 (Dipeptidyl peptidase-4)
ModalitySmall molecule
Therapeutic areaDiabetes
PhasePhase 3

Mechanism of action

By inhibiting DPP-4, gemigliptin prevents the degradation of glucagon-like peptide-1 (GLP-1) and glucose-dependent insulinotropic polypeptide (GIP), allowing these hormones to accumulate and enhance glucose-dependent insulin secretion. This mechanism reduces blood glucose levels in patients with type 2 diabetes while minimizing hypoglycemia risk since insulin secretion is glucose-dependent.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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