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DSM265 xmg

Medicines for Malaria Venture · Phase 2 active Small molecule

DSM265 is a dihydroorotate dehydrogenase (DHODH) inhibitor.

DSM265 is a dihydroorotate dehydrogenase (DHODH) inhibitor. Used for Malaria.

At a glance

Generic nameDSM265 xmg
SponsorMedicines for Malaria Venture
Drug classDHODH inhibitor
TargetDHODH
ModalitySmall molecule
Therapeutic areaInfectious Diseases
PhasePhase 2

Mechanism of action

DHODH is an enzyme involved in the de novo pyrimidine synthesis pathway. Inhibiting DHODH can lead to a decrease in the production of pyrimidine nucleotides, which are essential for DNA replication and cell division. This can be particularly effective against malaria parasites, which rely heavily on this pathway for survival.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results