PQP · Infectious Disease PQP is a quinolone-based antimalarial that inhibits parasite DNA gyrase and topoisomerase II, disrupting DNA replication in Plasmodium species.
Pyronaridine artesunate · Infectious Disease Pyronaridine artesunate is a fixed-dose combination antimalarial that kills malaria parasites through dual mechanisms: pyronaridine intercalates into parasite DNA while artesunate generates reactive oxygen species that damage parasite structures.
Phase 3 pipeline
Mefloquine plus artesunate · Infectious Disease This combination uses mefloquine (a quinoline antimalarial) and artesunate (an artemisinin derivative) to kill malaria parasites through complementary mechanisms that reduce drug resistance.
Phase 2 pipeline
DSM265 xmg · Infectious Diseases DSM265 is a dihydroorotate dehydrogenase (DHODH) inhibitor.