Last reviewed · How we verify

Larocaine (dimethocaine)

unknown active ✓ Verified May 2026

Larocaine (generic name: dimethocaine) is a dimethocaine drug. It is currently in unknown development.

Larocaine works by blocking the reuptake of certain neurotransmitters, such as norepinephrine, serotonin, and dopamine, in the brain.

Dimethocaine, also known as larocaine, is a compound with a stimulatory effect that resembles cocaine but is reportedly less potent. It is listed as a legal cocaine replacement in some countries and is addictive due to its stimulation of the reward pathway in the brain.

At a glance

Generic namedimethocaine
Drug classdimethocaine
Therapeutic areaNeuroscience
Phaseunknown

Mechanism of action

Imagine your brain is a city with many different streets and intersections. Neurotransmitters are like cars that carry messages between different parts of the city. Larocaine helps keep these cars on the streets longer, allowing them to deliver their messages more effectively.

Approved indications

No approved indications tracked.

Common side effects

No common side effects on file.

Competitive intelligence

For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:

Frequently asked questions about Larocaine

What is Larocaine?

Larocaine (dimethocaine) is a dimethocaine drug.

How does Larocaine work?

Larocaine works by blocking the reuptake of certain neurotransmitters, such as norepinephrine, serotonin, and dopamine, in the brain.

What is the generic name of Larocaine?

dimethocaine is the generic (nonproprietary) name of Larocaine.

What drug class is Larocaine in?

Larocaine belongs to the dimethocaine class. See all dimethocaine drugs at /class/dimethocaine.

What development phase is Larocaine in?

Larocaine is in unknown.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing