Last reviewed · How we verify
Difluprednate Ophthalmic
Difluprednate Ophthalmic is a Corticosteroid Small molecule drug developed by Thomas M. Lietman. It is currently FDA-approved for Post-operative inflammation following ocular surgery, Anterior uveitis, Inflammatory conditions of the anterior segment of the eye.
Difluprednate is a potent corticosteroid that suppresses inflammatory and immune responses in the eye by binding to glucocorticoid receptors.
Difluprednate is a potent corticosteroid that suppresses inflammatory and immune responses in the eye by binding to glucocorticoid receptors. Used for Post-operative inflammation following ocular surgery, Anterior uveitis, Inflammatory conditions of the anterior segment of the eye.
At a glance
| Generic name | Difluprednate Ophthalmic |
|---|---|
| Sponsor | Thomas M. Lietman |
| Drug class | Corticosteroid |
| Target | Glucocorticoid receptor |
| Modality | Small molecule |
| Therapeutic area | Ophthalmology |
| Phase | FDA-approved |
Mechanism of action
Difluprednate is a fluorinated prednisolone derivative designed for ophthalmic use with enhanced corneal penetration. It inhibits inflammatory mediators, reduces leukocyte infiltration, and suppresses immune cell activation in ocular tissues. The drug is particularly effective for post-operative inflammation and anterior uveitis due to its superior bioavailability in the anterior segment of the eye.
Approved indications
- Post-operative inflammation following ocular surgery
- Anterior uveitis
- Inflammatory conditions of the anterior segment of the eye
Common side effects
- Elevated intraocular pressure
- Posterior subcapsular cataract
- Ocular irritation or discomfort
- Secondary ocular infection
Key clinical trials
- Rose Bengal Electromagnetic Activation With Green Light for Infection Reduction II (PHASE3)
- A Study to Evaluate KRIYA-825 (VV-14295) in Adults With Geographic Atrophy Secondary to Age-related Macular Degeneration (PHASE1, PHASE2)
- Steroids and Cross-linking for Ulcer Treatment (PHASE3)
- Difluprednate vs. a Prednisolone Acetate - Phenylephrine on Post-operative Inflammation Following Cataract Surgery. (PHASE4)
- A Study of the Effect of Different Doses of Difluprednate Eye Drops on the Intraocular Pressure After Phacoemulsification (PHASE4)
- Clinical Investigation of the Dextenza 0.4mg Intracanalicular Insert Delivery System Used in Cataract Surgery (PHASE4)
- Topical Corticosteroid Use in Addition to Oral Antivirals for Prevention of Recurrence of Herpes Simplex Virus (HSV) Keratitis (PHASE4)
- Macular Edema Nepafenac vs. Difluprednate Uveitis Trial (PHASE4)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Difluprednate Ophthalmic CI brief — competitive landscape report
- Difluprednate Ophthalmic updates RSS · CI watch RSS
- Thomas M. Lietman portfolio CI
Frequently asked questions about Difluprednate Ophthalmic
What is Difluprednate Ophthalmic?
How does Difluprednate Ophthalmic work?
What is Difluprednate Ophthalmic used for?
Who makes Difluprednate Ophthalmic?
What drug class is Difluprednate Ophthalmic in?
What development phase is Difluprednate Ophthalmic in?
What are the side effects of Difluprednate Ophthalmic?
What does Difluprednate Ophthalmic target?
Related
- Drug class: All Corticosteroid drugs
- Target: All drugs targeting Glucocorticoid receptor
- Manufacturer: Thomas M. Lietman — full pipeline
- Therapeutic area: All drugs in Ophthalmology
- Indication: Drugs for Post-operative inflammation following ocular surgery
- Indication: Drugs for Anterior uveitis
- Indication: Drugs for Inflammatory conditions of the anterior segment of the eye
- Compare: Difluprednate Ophthalmic vs similar drugs
- Pricing: Difluprednate Ophthalmic cost, discount & access