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DHEA (1.0%)

EndoCeutics Inc. · Phase 3 active Small molecule

DHEA is a steroid hormone precursor that acts as a prohormone, being converted in peripheral tissues to testosterone and estrogen to restore hormonal balance.

DHEA is a steroid hormone precursor that acts as a prohormone, being converted in peripheral tissues to testosterone and estrogen to restore hormonal balance. Used for Moderate to severe dyspareunia (painful intercourse) due to menopause, Vaginal atrophy and related menopausal symptoms.

At a glance

Generic nameDHEA (1.0%)
Also known asPrasterone, Dehydroepiandrosterone
SponsorEndoCeutics Inc.
Drug classSteroid hormone / Prohormone
TargetAndrogen receptor, Estrogen receptor (via peripheral conversion)
ModalitySmall molecule
Therapeutic areaEndocrinology / Women's Health
PhasePhase 3

Mechanism of action

DHEA (dehydroepiandrosterone) is an endogenous steroid hormone that declines with age. When administered, it serves as a substrate for enzymatic conversion to active sex hormones (testosterone and estrogen) in target tissues. This mechanism aims to restore age-related hormonal deficiencies and improve symptoms associated with menopause and aging.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results