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Dapivirine Vaginal Ring-004
Dapivirine Vaginal Ring-004 is a Non-nucleoside reverse transcriptase inhibitor (NNRTI) Small molecule drug developed by International Partnership for Microbicides, Inc.. It is currently in Phase 3 development for HIV-1 prevention in women (pre-exposure prophylaxis). Also known as: TMC-120.
Dapivirine is a non-nucleoside reverse transcriptase inhibitor (NNRTI) that blocks HIV replication when released from a vaginal ring formulation.
Dapivirine is a non-nucleoside reverse transcriptase inhibitor (NNRTI) that blocks HIV replication when released from a vaginal ring formulation. Used for HIV-1 prevention in women (pre-exposure prophylaxis).
At a glance
| Generic name | Dapivirine Vaginal Ring-004 |
|---|---|
| Also known as | TMC-120 |
| Sponsor | International Partnership for Microbicides, Inc. |
| Drug class | Non-nucleoside reverse transcriptase inhibitor (NNRTI) |
| Target | HIV reverse transcriptase |
| Modality | Small molecule |
| Therapeutic area | Infectious Disease / Virology |
| Phase | Phase 3 |
Mechanism of action
Dapivirine inhibits HIV reverse transcriptase, preventing the virus from converting its RNA genome into DNA and integrating into host cells. The vaginal ring formulation provides sustained local and systemic drug delivery over several weeks, offering long-acting HIV prevention. This approach aims to provide women with a discreet, user-controlled contraceptive-like method for HIV pre-exposure prophylaxis (PrEP).
Approved indications
- HIV-1 prevention in women (pre-exposure prophylaxis)
Common side effects
- Vaginal irritation or discomfort
- Headache
- Vulvovaginal candidiasis
- Abnormal vaginal discharge
Key clinical trials
- Relative Bioavailability Trial of Dapivirine Ring-004 and Ring-008 (PHASE1)
- Safety and Pharmacokinetics of Dapivirine Vaginal Ring in Post-menopausal Women (PHASE2)
- To Assess Continued Safety of and Adherence to the Dapivirine (25 mg) Vaginal Ring-004 in Healthy, HIV-negative Women (PHASE3)
- Functionality of Male Condoms With a Silicone Elastomer Vaginal RIng (PHASE1)
- DDI Potential: Dapivirine Vaginal Ring and Miconazole Nitrate (PHASE1)
- A Trial In Healthy HIV-Negative Women To Assess The Effect Of Menses And Tampon Use On The Pharmacokinetics Of Dapivirine, Delivered By Dapivirine Vaginal Ring-004, Containing 25 Mg Of Dapivirine (PHASE1)
- To Assess the Drug-drug Interaction Potential Between Dapivirine Vaginal Ring-004, Containing 25 mg of Dapivirine, and Clotrimazole 10 mg/g (1%) (PHASE1)
- Expanded Use PK of Dapivirine Vaginal Ring (PHASE1)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Dapivirine Vaginal Ring-004 CI brief — competitive landscape report
- Dapivirine Vaginal Ring-004 updates RSS · CI watch RSS
- International Partnership for Microbicides, Inc. portfolio CI
Frequently asked questions about Dapivirine Vaginal Ring-004
What is Dapivirine Vaginal Ring-004?
How does Dapivirine Vaginal Ring-004 work?
What is Dapivirine Vaginal Ring-004 used for?
Who makes Dapivirine Vaginal Ring-004?
Is Dapivirine Vaginal Ring-004 also known as anything else?
What drug class is Dapivirine Vaginal Ring-004 in?
What development phase is Dapivirine Vaginal Ring-004 in?
What are the side effects of Dapivirine Vaginal Ring-004?
What does Dapivirine Vaginal Ring-004 target?
Related
- Drug class: All Non-nucleoside reverse transcriptase inhibitor (NNRTI) drugs
- Target: All drugs targeting HIV reverse transcriptase
- Manufacturer: International Partnership for Microbicides, Inc. — full pipeline
- Therapeutic area: All drugs in Infectious Disease / Virology
- Indication: Drugs for HIV-1 prevention in women (pre-exposure prophylaxis)
- Also known as: TMC-120
- Compare: Dapivirine Vaginal Ring-004 vs similar drugs
- Pricing: Dapivirine Vaginal Ring-004 cost, discount & access