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Dalteparin (Fragmin)

M.D. Anderson Cancer Center · FDA-approved active Small molecule Under review Quality 0/100

Dalteparin (Fragmin) is a Low-molecular-weight heparin (LMWH) Small molecule drug developed by M.D. Anderson Cancer Center. It is currently FDA-approved for Thromboprophylaxis in patients undergoing abdominal surgery, Thromboprophylaxis in patients with restricted mobility during acute illness, Treatment of acute deep vein thrombosis.

Dalteparin is a low-molecular-weight heparin that inhibits blood coagulation by enhancing the activity of antithrombin III against factor Xa and thrombin.

Dalteparin, also known as Fragmin, is an oligosaccharide antithrombin-III activator used to treat various conditions, including venous thromboembolism and pulmonary thromboembolisms. It is administered subcutaneously, either through traditional injections or via once-weekly subcutaneous ports, and its effectiveness can be monitored through point-of-care testing methods such as anti-Xa activity point-of-care testing.

At a glance

Generic nameDalteparin (Fragmin)
SponsorM.D. Anderson Cancer Center
Drug classLow-molecular-weight heparin (LMWH)
TargetAntithrombin III (indirect target); Factor Xa and Factor IIa (thrombin)
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved

Mechanism of action

Dalteparin binds to and potentiates antithrombin III, a natural anticoagulant, leading to inactivation of activated clotting factors, particularly factor Xa and to a lesser extent thrombin. This prevents thrombus formation and is used for thromboprophylaxis and treatment of thromboembolic disorders. It has a more predictable pharmacokinetic profile and longer half-life compared to unfractionated heparin.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Dalteparin (Fragmin)

What is Dalteparin (Fragmin)?

Dalteparin (Fragmin) is a Low-molecular-weight heparin (LMWH) drug developed by M.D. Anderson Cancer Center, indicated for Thromboprophylaxis in patients undergoing abdominal surgery, Thromboprophylaxis in patients with restricted mobility during acute illness, Treatment of acute deep vein thrombosis.

How does Dalteparin (Fragmin) work?

Dalteparin is a low-molecular-weight heparin that inhibits blood coagulation by enhancing the activity of antithrombin III against factor Xa and thrombin.

What is Dalteparin (Fragmin) used for?

Dalteparin (Fragmin) is indicated for Thromboprophylaxis in patients undergoing abdominal surgery, Thromboprophylaxis in patients with restricted mobility during acute illness, Treatment of acute deep vein thrombosis, Treatment of pulmonary embolism, Unstable angina and non-ST-segment elevation myocardial infarction.

Who makes Dalteparin (Fragmin)?

Dalteparin (Fragmin) is developed and marketed by M.D. Anderson Cancer Center (see full M.D. Anderson Cancer Center pipeline at /company/m-d-anderson-cancer-center).

What drug class is Dalteparin (Fragmin) in?

Dalteparin (Fragmin) belongs to the Low-molecular-weight heparin (LMWH) class. See all Low-molecular-weight heparin (LMWH) drugs at /class/low-molecular-weight-heparin-lmwh.

What development phase is Dalteparin (Fragmin) in?

Dalteparin (Fragmin) is FDA-approved (marketed).

What are the side effects of Dalteparin (Fragmin)?

Common side effects of Dalteparin (Fragmin) include Bleeding, Thrombocytopenia, Injection site hematoma, Elevated liver enzymes.

What does Dalteparin (Fragmin) target?

Dalteparin (Fragmin) targets Antithrombin III (indirect target); Factor Xa and Factor IIa (thrombin) and is a Low-molecular-weight heparin (LMWH).

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing