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Chlorhexidine gluconate at 0.12%

Universidad de Guanajuato · Phase 3 active Small molecule

Chlorhexidine gluconate is a broad-spectrum antimicrobial agent that disrupts bacterial cell membranes and denatures proteins, leading to rapid bactericidal and bacteriostatic effects.

Chlorhexidine gluconate is a broad-spectrum antimicrobial agent that disrupts bacterial cell membranes and denatures proteins, leading to rapid bactericidal and bacteriostatic effects. Used for Oral rinse for reduction of plaque and gingivitis, Antimicrobial oral care in Phase 3 development.

At a glance

Generic nameChlorhexidine gluconate at 0.12%
SponsorUniversidad de Guanajuato
Drug classAntimicrobial agent / Antiseptic
TargetBacterial cell membrane
ModalitySmall molecule
Therapeutic areaInfectious Disease / Oral Health
PhasePhase 3

Mechanism of action

Chlorhexidine is a cationic biguanide that binds to negatively charged bacterial cell membranes, causing leakage of cellular contents and protein denaturation. At the 0.12% concentration, it exhibits both bactericidal activity against gram-positive and gram-negative bacteria and some antifungal properties. It is commonly used as an oral rinse and topical antiseptic due to its broad-spectrum antimicrobial activity and low systemic absorption.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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