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Carbamazepine (Tegretol)
Carbamazepine (Tegretol) is a Anticonvulsant; sodium channel blocker Small molecule drug developed by Korean Epilepsy Society. It is currently FDA-approved for Epilepsy (generalized tonic-clonic and partial seizures), Trigeminal neuralgia, Bipolar disorder (acute mania and maintenance). Also known as: Tegretol, Carbamazepine (Tegretol-XR) placebo..
Carbamazepine stabilizes neuronal membranes and reduces repetitive neuronal firing by blocking voltage-gated sodium channels.
Carbamazepine stabilizes neuronal membranes and reduces repetitive neuronal firing by blocking voltage-gated sodium channels. Used for Epilepsy (generalized tonic-clonic and partial seizures), Trigeminal neuralgia, Bipolar disorder (acute mania and maintenance).
At a glance
| Generic name | Carbamazepine (Tegretol) |
|---|---|
| Also known as | Tegretol, Carbamazepine (Tegretol-XR) placebo. |
| Sponsor | Korean Epilepsy Society |
| Drug class | Anticonvulsant; sodium channel blocker |
| Target | Voltage-gated sodium channels |
| Modality | Small molecule |
| Therapeutic area | Neurology |
| Phase | FDA-approved |
Mechanism of action
The drug binds to inactivated sodium channels in the brain, preventing their reopening and thereby reducing the frequency of action potentials. This membrane-stabilizing effect suppresses abnormal electrical activity in the central nervous system, making it effective for controlling seizures and neuropathic pain. It also has mild anticholinergic and antidiuretic properties.
Approved indications
- Epilepsy (generalized tonic-clonic and partial seizures)
- Trigeminal neuralgia
- Bipolar disorder (acute mania and maintenance)
- Neuropathic pain
Common side effects
- Dizziness
- Ataxia
- Diplopia
- Nausea
- Rash (including Stevens-Johnson syndrome)
- Hyponatremia
- Agranulocytosis
- Hepatotoxicity
Key clinical trials
- A Study to Learn if Multiple Doses of the Study Medicine Called Carbamazepine Changes How the Body Processes the Other Study Medicine PF-07248144 (PHASE1)
- Pharmacological Mechanisms of Low-intensity Focused Ultrasound for Motor Cortex Neuroplasticity (EARLY_PHASE1)
- A Drug-Drug Interaction Study of Carbamazepine and Opevesostat (MK-5684) in Healthy Adult Male Participants (MK-5684-012) (PHASE1)
- A Study of Ponesimod in Healthy Adult Participants (PHASE1)
- A Drug-drug Interaction Study of S-892216 Coadministered With Carbamazepime to Healthy Adult Participants (PHASE1)
- Comparison of Oxcarbazepine Versus Carbamazepine in the Management of Trigeminal Neuralgia (PHASE4)
- A Trial to Evaluate the Effects of Itraconazole and Carbamazepine on the Pharmacokinetics of Emraclidine and of Emraclidine on the Pharmacokinetics of Metformin in Healthy Adult Participants (PHASE1)
- Longitudinal Comparative Effectiveness of Bipolar Disorder Therapies
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Carbamazepine (Tegretol) CI brief — competitive landscape report
- Carbamazepine (Tegretol) updates RSS · CI watch RSS
- Korean Epilepsy Society portfolio CI
Frequently asked questions about Carbamazepine (Tegretol)
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Related
- Drug class: All Anticonvulsant; sodium channel blocker drugs
- Target: All drugs targeting Voltage-gated sodium channels
- Manufacturer: Korean Epilepsy Society — full pipeline
- Therapeutic area: All drugs in Neurology
- Indication: Drugs for Epilepsy (generalized tonic-clonic and partial seizures)
- Indication: Drugs for Trigeminal neuralgia
- Indication: Drugs for Bipolar disorder (acute mania and maintenance)
- Also known as: Tegretol, Carbamazepine (Tegretol-XR) placebo.
- Compare: Carbamazepine (Tegretol) vs similar drugs
- Pricing: Carbamazepine (Tegretol) cost, discount & access