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Benadryl demand

University of Pennsylvania · FDA-approved active Small molecule

Benadryl (diphenhydramine) is a first-generation antihistamine that blocks H1 histamine receptors to reduce allergic and inflammatory responses.

Benadryl (diphenhydramine) is a first-generation antihistamine that blocks H1 histamine receptors to reduce allergic and inflammatory responses. Used for Allergic reactions and urticaria, Pruritus, Allergic rhinitis.

At a glance

Generic nameBenadryl demand
Also known asDiphenhydramine Hcl, Aler-Dryl, Banophen, Ben Tann, Bromanate AF
SponsorUniversity of Pennsylvania
Drug classFirst-generation H1 antihistamine
TargetH1 histamine receptor
ModalitySmall molecule
Therapeutic areaAllergy/Immunology
PhaseFDA-approved

Mechanism of action

Diphenhydramine competitively antagonizes H1 histamine receptors on various tissues, preventing histamine-mediated effects such as itching, urticaria, and allergic reactions. It also has anticholinergic properties that contribute to its sedating effects. The drug crosses the blood-brain barrier readily, which accounts for its central nervous system effects including drowsiness.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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