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Anoro® Ellipta®

AstraZeneca · FDA-approved active Small molecule

Anoro Ellipta combines a long-acting beta-2 agonist and a long-acting muscarinic antagonist to relax airway smooth muscle and improve airflow in chronic obstructive pulmonary disease.

Anoro® Ellipta® is a fixed-dose combination inhaler containing indacaterol maleate and glycopyrronium bromide, indicated for COPD. It has completed several clinical trials, demonstrating efficacy and safety. Despite no FDA label, it remains a key treatment option in COPD management.

At a glance

Generic nameAnoro® Ellipta®
Also known asAnoro® - Umeclidinium/Vilanterol, Ellipta® - Device, umeclidinium + vilanterol
SponsorAstraZeneca
Drug classLong-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination)
TargetBeta-2 adrenergic receptor and M3 muscarinic acetylcholine receptor
ModalitySmall molecule
Therapeutic areaRespiratory / Pulmonology
PhaseFDA-approved

Mechanism of action

The drug contains umeclidinium (a long-acting muscarinic antagonist) and vilanterol (a long-acting beta-2 agonist). These two bronchodilators work synergistically through different pathways: the beta-2 agonist increases cAMP to relax smooth muscle, while the muscarinic antagonist blocks acetylcholine-mediated bronchoconstriction. Together they provide sustained bronchodilation and improved lung function in COPD patients.

Approved indications

Common side effects

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