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AKR1C3-activated Prodrug AST-3424

SWOG Cancer Research Network · Phase 1 active Small molecule

Activates AKR1C3

Activates AKR1C3 Used for Solid tumors.

At a glance

Generic nameAKR1C3-activated Prodrug AST-3424
Also known asAKR1C3-activated Prodrug OBI-3424, AKR1C3-activated Prodrug TH-3424, Aldo-keto Reductase 1c3-activated Prodrug OBI-3424, AST-3424, OBI 3424
SponsorSWOG Cancer Research Network
Drug classProdrug
TargetAKR1C3
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 1

Mechanism of action

AST-3424 is a prodrug that is converted into an active form that activates the AKR1C3 enzyme.

Approved indications

Common side effects

No common side effects on file.

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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