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AJG555

EA Pharma Co., Ltd. · Phase 3 active Small molecule

AJG555 is a guanylate cyclase-C (GC-C) agonist that increases intracellular cGMP to promote fluid secretion and accelerate intestinal transit.

AJG555 is a guanylate cyclase-C (GC-C) agonist that increases intracellular cGMP to promote fluid secretion and accelerate intestinal transit. Used for Irritable bowel syndrome with constipation (IBS-C), Chronic idiopathic constipation (CIC).

At a glance

Generic nameAJG555
SponsorEA Pharma Co., Ltd.
Drug classGuanylate cyclase-C agonist
TargetGC-C (guanylate cyclase-C)
ModalitySmall molecule
Therapeutic areaGastroenterology
PhasePhase 3

Mechanism of action

By activating guanylate cyclase-C receptors on intestinal epithelial cells, AJG555 increases cyclic GMP levels, which triggers chloride and bicarbonate secretion into the intestinal lumen and enhances intestinal motility. This mechanism promotes stool passage and is designed to treat functional gastrointestinal disorders characterized by constipation or reduced intestinal transit.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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