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Vegf Trap (AFLIBERCEPT)
Aflibercept, also known as Vegf Trap, is a vascular endothelial growth factor inhibitor developed by Regeneron Pharmaceuticals. It works by binding to vascular endothelial growth factor A, preventing its interaction with its receptor and thereby inhibiting angiogenesis. Aflibercept is approved to treat various eye conditions, including macular edema and age-related macular degeneration, as well as metastatic colorectal cancer. It is a small molecule drug that has been commercially available since 2011. Key safety considerations include potential increased risk of hypertension, proteinuria, and gastrointestinal perforation.
At a glance
| Generic name | AFLIBERCEPT |
|---|---|
| Sponsor | Regeneron |
| Drug class | Vascular Endothelial Growth Factor Inhibitor |
| Target | Vascular endothelial growth factor A |
| Modality | Recombinant protein |
| Therapeutic area | Oncology |
| Phase | FDA-approved |
| First approval | 2011 |
| Annual revenue | 9800 |
Approved indications
- Branch retinal vein occlusion with macular edema
- Central retinal vein occlusion with macular edema
- Exudative age-related macular degeneration
- Macular edema due to diabetes mellitus
- Metastasis from malignant tumor of colon
- Neovascular glaucoma
- Retinopathy of prematurity
Common side effects
- Leukopenia
- Neutropenia
- Diarrhea
- Proteinuria
- AST increased
- Stomatitis
- Fatigue
- Thrombocytopenia
- ALT increased
- Hypertension
- Weight decreased
- Decreased appetite
Key clinical trials
- Testing the PD-1 Antibody, MK3475, Given With Ziv-aflibercept in Patients With Advanced Cancer (PHASE1)
- A Clinical Trial of EYE201/MK-8748 in People With Macular Degeneration (MK-8748-003) (PHASE2,PHASE3)
- Extension Study to Evaluate the Long-Term Outcomes of Pediatric Patients Who Received Treatment for Retinopathy of Prematurity in the VGFTe-ROP-1920 Study (Acronym: Butterfleye Next)
- 4D-150 in Patients With Macular Neovascularization Secondary to Age-Related Macular Degeneration (PHASE3)
- A Clinical Study of QL1207H Injection Versus Aflibercept for Neovascular Age-related Macular Degeneration (PHASE3)
- Clinical Study to Compare Efficacy and Safety of AVT29 and Eylea HD in Participants With Diabetic Macular Edema (PHASE3)
- Efficacy and Safety Study of Ixoberogene Soroparvovec (Ixo-vec) in Participants With Neovascular Age-related Macular Degeneration (AQUARIUS) (PHASE3)
- An Observational Study to Collect Data on How Aflibercept (Eylea) Given Using a Paediatric Dosing Device is Used in Preterm Babies With Retinopathy of Prematurity in the United Kingdom (UK)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| FDA label | Mechanism, indications, dosing, boxed warnings, drug interactions |
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
| SEC EDGAR | Revenue + earnings |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Vegf Trap CI brief — competitive landscape report
- Vegf Trap updates RSS · CI watch RSS
- Regeneron portfolio CI