nonsteroidal antiandrogen
This page covers all nonsteroidal antiandrogen drugs tracked by Drug Landscape: marketed products and active clinical-stage compounds, targeting androgen receptor, Androgen receptor, Androgen receptor; GnRH receptor (depending on specific agents used).
Targets
androgen receptor · Androgen receptor · Androgen receptor; GnRH receptor (depending on specific agents used)
Phase 3 pipeline (4)
- Placebo of Darolutamide · Association Pour La Recherche des Thérapeutiques Innovantes en Cancérologie · Oncology
Darolutamide is a nonsteroidal antiandrogen that competitively inhibits the action of androgens, such as testosterone and dihydrotestosterone, at their receptor sites in various tissues. - Long-term course of antiandrogen drugs · The First Affiliated Hospital with Nanjing Medical University · Oncology
Antiandrogen drugs block the effects of androgens (male hormones) by inhibiting androgen receptor signaling. - Adjuvant Androgen-Deprivation Therapy · National Taiwan University Hospital · Oncology
Adjuvant androgen-deprivation therapy suppresses testosterone production to inhibit the growth of hormone-sensitive prostate cancer cells after primary treatment. - Standard Darolutamide · Jena University Hospital · Oncology
Darolutamide is a nonsteroidal antiandrogen that competitively inhibits the action of androgens, such as testosterone and dihydrotestosterone, at their receptor sites in various tissues.
Phase 2 pipeline (1)
- Bicalutamide Oral Product · Gynaecologisch Oncologisch Centrum Zuid · Oncology
Bicalutamide is a nonsteroidal antiandrogen that inhibits the action of androgens.
Patent intelligence
- antiandrogen patent landscape — aggregated cliff calendar, attackable patents, originator estates