What are Alpha-1A adrenergic receptor antagonist drugs?

Alpha-1A adrenergic receptor antagonist drugs are pharmacologic agents that share a common mechanism (typically targeting Alpha-1A adrenergic receptor). 2 are currently marketed, with 4 more in clinical development.

What are the marketed Alpha-1A adrenergic receptor antagonist drugs?

Marketed Alpha-1A adrenergic receptor antagonist drugs include Tamsulosin BID, Tamsulosine Arrow LP.

Alpha-1A adrenergic receptor antagonist

2 marketed 4 in Phase 3

This page covers all Alpha-1A adrenergic receptor antagonist drugs tracked by Drug Landscape: marketed products and active clinical-stage compounds, targeting Alpha-1A adrenergic receptor.

Targets

Alpha-1A adrenergic receptor

Marketed (2)

Tamsulosin BID · Gundersen Lutheran Medical Foundation · Urology
Tamsulosin is an alpha-1A adrenergic receptor antagonist that relaxes smooth muscle in the prostate and bladder neck to improve urinary flow.
Tamsulosine Arrow LP · Pierre Fabre Medicament · Urology
Tamsulosin is an alpha-1A adrenergic receptor antagonist that relaxes smooth muscle in the prostate and bladder neck to improve urinary flow.

Phase 3 pipeline (4)

Uroxatrol (drug) · New York Prostate Institute · Urology
Uroxatrol is an alpha-1A adrenergic receptor antagonist that relaxes smooth muscle in the prostate and bladder neck to improve urinary flow.
Omnic Ocas · EMS · Urology
Omnic Ocas is a once-daily oral formulation of tamsulosin that selectively blocks alpha-1A adrenergic receptors in the prostate and bladder neck to relieve urinary obstruction.
Disintegrating placebo tamsulosin tablet · GlaxoSmithKline · Urology
Tamsulosin is an alpha-1A adrenergic receptor antagonist that relaxes smooth muscle in the prostate and bladder neck to improve urinary flow.
Preventive administration of Rapaflo · Sir Mortimer B. Davis - Jewish General Hospital · Urology
Rapaflo (silodosin) is an alpha-1A adrenergic receptor antagonist that relaxes smooth muscle in the prostate and bladder neck to improve urinary flow.