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umeclidinium bromide and vilanterol trifenatate — Competitive Intelligence Brief
marketed
Long-acting muscarinic antagonist / Long-acting beta-2 agonist combination (LAMA/LABA)
M3 muscarinic receptor and beta-2 adrenergic receptor
Respiratory / Pulmonology
Small molecule
Live · refreshed every 30 min
Target snapshot
umeclidinium bromide and vilanterol trifenatate (umeclidinium bromide and vilanterol trifenatate) — Chiesi Farmaceutici S.p.A.. Umeclidinium is a long-acting muscarinic antagonist and vilanterol is a long-acting beta-2 agonist that together relax airway smooth muscle and improve airflow in chronic obstructive pulmonary disease.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| umeclidinium bromide and vilanterol trifenatate TARGET | umeclidinium bromide and vilanterol trifenatate | Chiesi Farmaceutici S.p.A. | marketed | Long-acting muscarinic antagonist / Long-acting beta-2 agonist combination (LAMA/LABA) | M3 muscarinic receptor and beta-2 adrenergic receptor | |
| GSK573719/VI 125/25 | GSK573719/VI 125/25 | GlaxoSmithKline | phase 3 | LAMA/LABA combination (long-acting muscarinic antagonist/long-acting beta-2 agonist) | M3 muscarinic receptor and beta-2 adrenergic receptor | |
| TIO/OLO | TIO/OLO | GlaxoSmithKline | marketed | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | Muscarinic M3 receptor and beta-2 adrenergic receptor | |
| UMEC/VI DPI | UMEC/VI DPI | GlaxoSmithKline | marketed | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | Muscarinic M3 receptor (umeclidinium); Beta-2 adrenergic receptor (vilanterol) | |
| Revefenacin 175 µg, Formoterol 20 µg | Revefenacin 175 µg, Formoterol 20 µg | University of Tennessee Graduate School of Medicine | marketed | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | M3 muscarinic receptor; beta-2 adrenergic receptor | |
| UMEC/VI | UMEC/VI | GlaxoSmithKline | marketed | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | Muscarinic M3 receptor; beta-2 adrenergic receptor | |
| Umeclidinium/Vilanterol 62.5/25 mcgs | Umeclidinium/Vilanterol 62.5/25 mcgs | National Institute of Respiratory Diseases, Mexico | marketed | Long-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA) | M3 muscarinic receptor; beta-2 adrenergic receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Long-acting muscarinic antagonist / Long-acting beta-2 agonist combination (LAMA/LABA) class)
- Chiesi Farmaceutici S.p.A. · 1 drug in this class
- Gary L. Pierce · 1 drug in this class
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Cite this brief
Drug Landscape (2026). umeclidinium bromide and vilanterol trifenatate — Competitive Intelligence Brief. https://druglandscape.com/ci/umeclidinium-bromide-and-vilanterol-trifenatate. Accessed 2026-05-18.
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