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UMEC/VI DPI

GlaxoSmithKline · FDA-approved active Small molecule

UMEC/VI is a combination of umeclidinium (a long-acting muscarinic antagonist) and vilanterol (a long-acting beta-2 agonist) that relaxes airway smooth muscle and improves airflow in chronic obstructive pulmonary disease.

UMEC/VI is a combination of umeclidinium (a long-acting muscarinic antagonist) and vilanterol (a long-acting beta-2 agonist) that relaxes airway smooth muscle and improves airflow in chronic obstructive pulmonary disease. Used for Chronic obstructive pulmonary disease (COPD) maintenance treatment.

At a glance

Generic nameUMEC/VI DPI
SponsorGlaxoSmithKline
Drug classLong-acting muscarinic antagonist / long-acting beta-2 agonist combination (LAMA/LABA)
TargetMuscarinic M3 receptor (umeclidinium); Beta-2 adrenergic receptor (vilanterol)
ModalitySmall molecule
Therapeutic areaRespiratory / Pulmonology
PhaseFDA-approved

Mechanism of action

Umeclidinium blocks muscarinic M3 receptors on airway smooth muscle, preventing acetylcholine-induced bronchoconstriction. Vilanterol activates beta-2 adrenergic receptors, promoting smooth muscle relaxation and bronchodilation. Together, these complementary mechanisms provide sustained bronchodilation over 24 hours.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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