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TR-701 FA — Competitive Intelligence Brief
phase 3
Oxazolidinone antibiotic
Bacterial 70S ribosome
Infectious Disease
Small molecule
Live · refreshed every 30 min
Target snapshot
TR-701 FA (TR-701 FA) — Trius Therapeutics LLC, a subsidiary of Merck & Co., Inc. (Rahway, New Jersey USA). TR-701 FA is a prodrug of TR-700 that inhibits bacterial protein synthesis by binding to the bacterial ribosome.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| TR-701 FA TARGET | TR-701 FA | Trius Therapeutics LLC, a subsidiary of Merck & Co., Inc. (Rahway, New Jersey USA) | phase 3 | Oxazolidinone antibiotic | Bacterial 70S ribosome | |
| Sivextro 200 milligrams Oral Tablet | Sivextro 200 milligrams Oral Tablet | Fundacion Clinic per a la Recerca Biomédica | marketed | Oxazolidinone antibiotic | Bacterial 70S ribosome (peptidyl transferase center) | |
| Synthomycine 5% | Synthomycine 5% | Barzilai Medical Center | marketed | Broad-spectrum antibiotic (chloramphenicol) | Bacterial 70S ribosome (peptidyl transferase) | |
| Linezolid (LZD) | Linezolid (LZD) | Wuhan Pulmonary Hospital | marketed | Oxazolidinone antibiotic | Bacterial 50S ribosomal subunit (23S rRNA) | |
| Tedizolid IV | Tedizolid IV | University of Southern California | marketed | Oxazolidinone antibiotic | Bacterial 50S ribosomal subunit | |
| Tedizolid PO | Tedizolid PO | University of Southern California | marketed | Oxazolidinone antibiotic | Bacterial 50S ribosomal subunit | |
| Linezolid Injectable Product | Linezolid Injectable Product | Fundacion Clinic per a la Recerca Biomédica | marketed | Oxazolidinone antibiotic | Bacterial 50S ribosomal subunit (23S rRNA) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Oxazolidinone antibiotic class)
- Fundacion Clinic per a la Recerca Biomédica · 2 drugs in this class
- University of Southern California · 2 drugs in this class
- Arpida AG · 2 drugs in this class
- Pfizer · 1 drug in this class
- Shenzhen Third People's Hospital · 1 drug in this class
- Trius Therapeutics LLC, a subsidiary of Merck & Co., Inc. (Rahway, New Jersey USA) · 1 drug in this class
- Wuhan Pulmonary Hospital · 1 drug in this class
- Clinica Universidad de Navarra, Universidad de Navarra · 1 drug in this class
- Merck Sharp & Dohme LLC · 1 drug in this class
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Cite this brief
Drug Landscape (2026). TR-701 FA — Competitive Intelligence Brief. https://druglandscape.com/ci/tr-701-fa. Accessed 2026-05-13.
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