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Tolterodine 6 — Competitive Intelligence Brief
marketed
Muscarinic receptor antagonist
M2 and M3 muscarinic receptors
Urology
Small molecule
Live · refreshed every 30 min
Target snapshot
Tolterodine 6 (Tolterodine 6) — KYU-SUNG LEE. Tolterodine is a muscarinic receptor antagonist that blocks acetylcholine signaling in the bladder to reduce involuntary contractions and urinary urgency.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Tolterodine 6 TARGET | Tolterodine 6 | KYU-SUNG LEE | marketed | Muscarinic receptor antagonist | M2 and M3 muscarinic receptors | |
| Tolterodine Tartrate ER | Tolterodine Tartrate ER | University of California, San Francisco | marketed | Muscarinic receptor antagonist | M2 and M3 muscarinic receptors | |
| Detrol LA | Detrol LA | Pfizer's Upjohn has merged with Mylan to form Viatris Inc. | marketed | Muscarinic receptor antagonist | M2 and M3 muscarinic acetylcholine receptors | |
| Atropine 1% | Atropine 1% | Massachusetts Eye and Ear Infirmary | marketed | Anticholinergic agent / Muscarinic receptor antagonist | Muscarinic acetylcholine receptors (M1-M5, primarily M3 in ocular tissue) | |
| Atropine Sulfate 0.04% Eye Drop | Atropine Sulfate 0.04% Eye Drop | Shanghai Eye Disease Prevention and Treatment Center | marketed | Anticholinergic agent / Muscarinic receptor antagonist | Muscarinic acetylcholine receptors (M1, M3, M5) | |
| Atropine sulfate eye drops 0.01% | Atropine sulfate eye drops 0.01% | Oupushifang Pharmaceutical Technology Co., Ltd. | phase 3 | Muscarinic receptor antagonist | Muscarinic acetylcholine receptors (M1, M3) | |
| Atropine Sulfate 02 | Atropine Sulfate 02 | LitePharmTech Co., Ltd. | phase 3 | Anticholinergic agent / Muscarinic receptor antagonist | Muscarinic acetylcholine receptors (M1-M5) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Muscarinic receptor antagonist class)
- KYU-SUNG LEE · 1 drug in this class
- Oupushifang Pharmaceutical Technology Co., Ltd. · 1 drug in this class
- Pfizer's Upjohn has merged with Mylan to form Viatris Inc. · 1 drug in this class
- R-Pharm · 1 drug in this class
- University of California, San Francisco · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Tolterodine 6 — Competitive Intelligence Brief. https://druglandscape.com/ci/tolterodine-6. Accessed 2026-05-16.
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