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Tienoridine — Competitive Intelligence Brief
phase 3
tinoridine
Adenosine receptor A1
Neuroscience
Small molecule
Live · refreshed every 30 min
Target snapshot
Tienoridine (TINORIDINE). Tienoridine works by binding to the adenosine receptor A1, which helps to reduce pain by modulating the activity of neurons.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Tienoridine TARGET | TINORIDINE | phase 3 | tinoridine | Adenosine receptor A1 | ||
| Neurontin | gabapentin | Generic (originally Parke-Davis/Pfizer) | marketed | Gabapentinoid (anticonvulsant/neuropathic pain agent) | Large neutral amino acids transporter small subunit 1, Adenosine receptor A1, Alpha-2A adrenergic receptor | 1993-12-30 |
| Oxtriphylline | choline theophyllinate | Warner Chilcott Llc | marketed | choline theophyllinate | Adenosine receptor A3, Alkaline phosphatase, tissue-nonspecific isozyme, Adenosine receptor A1 | 1981-01-01 |
| Predema | pamabrom | marketed | pamabrom | Adenosine receptor A1 | ||
| Aminophyllin | Aminophyllin | University of Padova | marketed | Adenosine receptor A3, Alkaline phosphatase, tissue-nonspecific isozyme, Adenosine receptor A1 | ||
| Theophyllin | Theophyllin | University of Bergen | marketed | Adenosine receptor A3, Alkaline phosphatase, tissue-nonspecific isozyme, Adenosine receptor A1 | ||
| Lexiscan | Lexiscan | Medical University of South Carolina | marketed | Adenosine receptor A3, Adenosine receptor A1, Adenosine receptor A2a |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (tinoridine class)
- · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Tienoridine — Competitive Intelligence Brief. https://druglandscape.com/ci/tinoridine. Accessed 2026-06-10.
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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing