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Technetium Tc99m Sestamibi — Competitive Intelligence Brief
marketed
Radiopharmaceutical imaging agent
Mitochondrial membrane potential
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Technetium Tc99m Sestamibi (Technetium Tc99m Sestamibi) — Lantheus Medical Imaging. Technetium Tc-99m sestamibi is a radiopharmaceutical that accumulates in mitochondria of viable myocardial cells, allowing visualization of myocardial perfusion and viability via nuclear imaging.
Comparator set (2 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Technetium Tc99m Sestamibi TARGET | Technetium Tc99m Sestamibi | Lantheus Medical Imaging | marketed | Radiopharmaceutical imaging agent | Mitochondrial membrane potential | |
| Technetium Tc99m Tetrofosmin injections | Technetium Tc99m Tetrofosmin injections | GE Healthcare | marketed | Myocardial perfusion imaging agent | Mitochondrial membrane potential in myocardial cells | |
| Tc99m sestamibi | Tc99m sestamibi | M.D. Anderson Cancer Center | marketed | Radiotracer / Diagnostic imaging agent | Mitochondrial membrane potential |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Radiopharmaceutical imaging agent class)
- Lantheus Medical Imaging · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Technetium Tc99m Sestamibi — Competitive Intelligence Brief. https://druglandscape.com/ci/technetium-tc99m-sestamibi. Accessed 2026-05-17.
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