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Rosiglitazone XR — Competitive Intelligence Brief
marketed
Thiazolidinedione (PPAR-γ agonist)
PPAR-γ (Peroxisome proliferator-activated receptor gamma)
Diabetes
Small molecule
Live · refreshed every 30 min
Target snapshot
Rosiglitazone XR (Rosiglitazone XR) — GlaxoSmithKline. Rosiglitazone is a thiazolidinedione that activates peroxisome proliferator-activated receptor gamma (PPAR-γ) to improve insulin sensitivity and reduce blood glucose in type 2 diabetes.
Comparator set (4 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Rosiglitazone XR TARGET | Rosiglitazone XR | GlaxoSmithKline | marketed | Thiazolidinedione (PPAR-γ agonist) | PPAR-γ (Peroxisome proliferator-activated receptor gamma) | |
| IMP Pioglitozone | IMP Pioglitozone | University of Nottingham | marketed | Thiazolidinedione (PPAR-γ agonist) | PPAR-γ (Peroxisome proliferator-activated receptor gamma) | |
| Pioglitazone Tablets | Pioglitazone Tablets | Peking Union Medical College Hospital | marketed | Thiazolidinedione (PPAR-γ agonist) | PPAR-γ (Peroxisome proliferator-activated receptor gamma) | |
| Pioglitazone, Rosiglitazone | Pioglitazone, Rosiglitazone | Korea University Anam Hospital | marketed | Thiazolidinedione (PPAR-γ agonist) | PPAR-γ (Peroxisome proliferator-activated receptor gamma) | |
| Pioglitazone rescue therapy | Pioglitazone rescue therapy | Merck Sharp & Dohme LLC | phase 3 | Thiazolidinedione (PPAR-γ agonist) | PPAR-γ (Peroxisome proliferator-activated receptor gamma) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Thiazolidinedione (PPAR-γ agonist) class)
- GlaxoSmithKline · 1 drug in this class
- Korea University Anam Hospital · 1 drug in this class
- Merck Sharp & Dohme LLC · 1 drug in this class
- Peking Union Medical College Hospital · 1 drug in this class
- University of Nottingham · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Rosiglitazone XR — Competitive Intelligence Brief. https://druglandscape.com/ci/rosiglitazone-xr. Accessed 2026-05-16.
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