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IMP Pioglitozone

University of Nottingham · FDA-approved active Small molecule

Pioglitazone activates peroxisome proliferator-activated receptor gamma (PPAR-γ) to improve insulin sensitivity and reduce blood glucose in type 2 diabetes.

Pioglitazone activates peroxisome proliferator-activated receptor gamma (PPAR-γ) to improve insulin sensitivity and reduce blood glucose in type 2 diabetes. Used for Type 2 diabetes mellitus.

At a glance

Generic nameIMP Pioglitozone
SponsorUniversity of Nottingham
Drug classThiazolidinedione (PPAR-γ agonist)
TargetPPAR-γ (Peroxisome proliferator-activated receptor gamma)
ModalitySmall molecule
Therapeutic areaDiabetes
PhaseFDA-approved

Mechanism of action

As a thiazolidinedione, pioglitazone binds to PPAR-γ in adipose tissue and muscle, enhancing insulin-mediated glucose uptake and reducing hepatic glucose production. This mechanism addresses insulin resistance, the underlying pathophysiology of type 2 diabetes, rather than stimulating insulin secretion directly.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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