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Regadenoson peripheral - peripheral — Competitive Intelligence Brief
phase 3
Adenosine A2A receptor agonist
Adenosine A2A receptor
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Regadenoson peripheral - peripheral (Regadenoson peripheral - peripheral) — Lokien van Nunen. Regadenoson is an adenosine A2A receptor agonist that causes peripheral vasodilation to increase blood flow, used as a pharmacologic stress agent for cardiac imaging.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Regadenoson peripheral - peripheral TARGET | Regadenoson peripheral - peripheral | Lokien van Nunen | phase 3 | Adenosine A2A receptor agonist | Adenosine A2A receptor | |
| Regadenoson (Lexiscan) | Regadenoson (Lexiscan) | Brigham and Women's Hospital | marketed | Adenosine A2A receptor agonist | Adenosine A2A receptor | |
| Regadenoson myocardial perfusion imaging | Regadenoson myocardial perfusion imaging | University of Colorado, Denver | marketed | Adenosine A2A receptor agonist | Adenosine A2A receptor | |
| Regadenoson MRI myocardial blood flow | Regadenoson MRI myocardial blood flow | University of Colorado, Denver | marketed | Adenosine A2A receptor agonist | Adenosine A2A receptor | |
| Istradefylline (KW-6002) | Istradefylline (KW-6002) | Kyowa Kirin, Inc. | phase 3 | Adenosine A2A receptor antagonist | Adenosine A2A receptor | |
| Regadenoson peripheral - central | Regadenoson peripheral - central | Lokien van Nunen | phase 3 | Adenosine A2A receptor agonist | Adenosine A2A receptor | |
| Pharmacological stress agents | Pharmacological stress agents | GE Healthcare | phase 3 | Cardiac stress agents | Adenosine A2A receptor (adenosine); dopamine and beta-adrenergic receptors (dobutamine); adenosine A2A receptor (regadenoson) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Adenosine A2A receptor agonist class)
- Lokien van Nunen · 2 drugs in this class
- University of Colorado, Denver · 2 drugs in this class
- Brigham and Women's Hospital · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Regadenoson peripheral - peripheral — Competitive Intelligence Brief. https://druglandscape.com/ci/regadenoson-peripheral-peripheral. Accessed 2026-05-13.
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