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Regadenoson central - peripheral — Competitive Intelligence Brief
phase 3
Adenosine receptor agonist
A2A receptor
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Regadenoson central - peripheral (Regadenoson central - peripheral) — Lokien van Nunen. Regadenoson central - peripheral acts as an adenosine A2A receptor agonist.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Regadenoson central - peripheral TARGET | Regadenoson central - peripheral | Lokien van Nunen | phase 3 | Adenosine receptor agonist | A2A receptor | |
| Regadenoson MRI myocardial blood flow | Regadenoson MRI myocardial blood flow | University of Colorado, Denver | marketed | Adenosine A2A receptor agonist | Adenosine A2A receptor | |
| SG | SG | Arcus Biosciences, Inc. | marketed | Adenosine 2A receptor antagonist | A2A receptor (adenosine 2A receptor) | |
| Regadenoson myocardial perfusion imaging | Regadenoson myocardial perfusion imaging | University of Colorado, Denver | marketed | Adenosine A2A receptor agonist | Adenosine A2A receptor | |
| Regadenoson (Lexiscan) | Regadenoson (Lexiscan) | Brigham and Women's Hospital | marketed | Adenosine A2A receptor agonist | Adenosine A2A receptor | |
| AD109 | AD109 | Apnimed | phase 3 | Adenosine A2A receptor antagonist | Adenosine A2A receptor | |
| Regadenoson central -central | Regadenoson central -central | Lokien van Nunen | phase 3 | A2A receptor agonist | A2A receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Adenosine receptor agonist class)
- Inotek Pharmaceuticals Corporation · 1 drug in this class
- Lokien van Nunen · 1 drug in this class
- Pfizer Inc. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Regadenoson central - peripheral — Competitive Intelligence Brief. https://druglandscape.com/ci/regadenoson-central-peripheral. Accessed 2026-05-14.
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