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Preemptive Analgesia Of Dexmedetomidine — Competitive Intelligence Brief
marketed
Alpha-2 adrenergic agonist
Alpha-2 adrenergic receptor
Anesthesia and Pain Management
Small molecule
Live · refreshed every 30 min
Target snapshot
Preemptive Analgesia Of Dexmedetomidine (Preemptive Analgesia Of Dexmedetomidine) — China International Neuroscience Institution. Dexmedetomidine is a selective alpha-2 adrenergic agonist that reduces pain perception and provides analgesia through central nervous system effects.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Preemptive Analgesia Of Dexmedetomidine TARGET | Preemptive Analgesia Of Dexmedetomidine | China International Neuroscience Institution | marketed | Alpha-2 adrenergic agonist | Alpha-2 adrenergic receptor | |
| Nebulized lidocaine and dexmedetomidine | Nebulized lidocaine and dexmedetomidine | Ain Shams University | marketed | Local anesthetic and sedative-analgesic combination | Voltage-gated sodium channels (lidocaine); alpha-2 adrenergic receptors (dexmedetomidine) | |
| Oxymetazoline gel | Oxymetazoline gel | RDD Pharma Ltd | marketed | Alpha-2 adrenergic agonist | Alpha-2 adrenergic receptor | |
| ketamine- dexmeditomidine admixure | ketamine- dexmeditomidine admixure | Kasr El Aini Hospital | marketed | Dissociative anesthetic with alpha-2 adrenergic agonist | NMDA receptor (ketamine); alpha-2 adrenergic receptor (dexmedetomidine) | |
| brimonidine 0.1% (Alphagan® P) | brimonidine 0.1% (Alphagan® P) | Allergan | marketed | Alpha-2 adrenergic receptor agonist | Alpha-2 adrenergic receptor | |
| Dexmedetomidine for sedation | Dexmedetomidine for sedation | Southeast University, China | marketed | Alpha-2 adrenergic receptor agonist | Alpha-2 adrenergic receptor | |
| transdermal clonidine | transdermal clonidine | Peking University People's Hospital | marketed | Alpha-2 adrenergic agonist | Alpha-2 adrenergic receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Alpha-2 adrenergic agonist class)
- USWM, LLC (dba US WorldMeds) · 2 drugs in this class
- China International Neuroscience Institution · 1 drug in this class
- Icahn School of Medicine at Mount Sinai · 1 drug in this class
- Eye Therapies, LLC · 1 drug in this class
- Galderma R&D · 1 drug in this class
- Guangzhou Women and Children's Medical Center · 1 drug in this class
- Derm Research, PLLC · 1 drug in this class
- Irmandade da Santa Casa de Misericordia de Sao Paulo · 1 drug in this class
- KK Women's and Children's Hospital · 1 drug in this class
- American University of Beirut Medical Center · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Preemptive Analgesia Of Dexmedetomidine — Competitive Intelligence Brief. https://druglandscape.com/ci/preemptive-analgesia-of-dexmedetomidine. Accessed 2026-05-17.
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