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Olodaterol-Tiotropium — Competitive Intelligence Brief
marketed
Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination)
Beta-2 adrenergic receptor; M3 muscarinic receptor
Respiratory / Pulmonology
Small molecule
Live · refreshed every 30 min
Target snapshot
Olodaterol-Tiotropium (Olodaterol-Tiotropium) — Fraunhofer-Institute of Toxicology and Experimental Medicine. Olodaterol-Tiotropium is a fixed-dose combination of a long-acting beta-2 agonist (olodaterol) and a long-acting muscarinic antagonist (tiotropium) that work synergistically to relax airway smooth muscle and improve airflow.
Comparator set (5 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Olodaterol-Tiotropium TARGET | Olodaterol-Tiotropium | Fraunhofer-Institute of Toxicology and Experimental Medicine | marketed | Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) | Beta-2 adrenergic receptor; M3 muscarinic receptor | |
| Vilanterol and Umeclidinium Bromide | Vilanterol and Umeclidinium Bromide | Samsung Medical Center | marketed | Long-acting beta-2 agonist / Long-acting muscarinic antagonist combination (LABA/LAMA) | Beta-2 adrenergic receptor; M3 muscarinic receptor | |
| FF/GW642444 Inhalation Powder | FF/GW642444 Inhalation Powder | GlaxoSmithKline | phase 3 | Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) | Beta-2 adrenergic receptor; M3 muscarinic receptor | |
| Anoro® Ellipta® | Anoro® Ellipta® | AstraZeneca | marketed | Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) | Beta-2 adrenergic receptor and M3 muscarinic acetylcholine receptor | |
| Indacaterol/glycopyrronium | Indacaterol/glycopyrronium | Orion Corporation, Orion Pharma | marketed | Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) | Beta-2 adrenergic receptor; M3 muscarinic acetylcholine receptor | |
| indacaterol/glycopyrronium 110/50 Breezhaler® | indacaterol/glycopyrronium 110/50 Breezhaler® | Wouter H. van Geffen | marketed | Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) | Beta-2 adrenergic receptor; Muscarinic M3 acetylcholine receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) class)
- AstraZeneca · 1 drug in this class
- Fraunhofer-Institute of Toxicology and Experimental Medicine · 1 drug in this class
- GlaxoSmithKline · 1 drug in this class
- Orion Corporation, Orion Pharma · 1 drug in this class
- Wouter H. van Geffen · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Olodaterol-Tiotropium — Competitive Intelligence Brief. https://druglandscape.com/ci/olodaterol-tiotropium. Accessed 2026-05-16.
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