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nicotine acid — Competitive Intelligence Brief
phase 3
lipid-regulating agent
GPR109A
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
nicotine acid (nicotine acid) — GWT-TUD GmbH. Nicotine acid, also known as niacin, primarily functions by reducing the production of very-low-density lipoprotein (VLDL) and low-density lipoprotein (LDL) cholesterol in the liver.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| nicotine acid TARGET | nicotine acid | GWT-TUD GmbH | phase 3 | lipid-regulating agent | GPR109A | |
| Nicotinic acid (niacin) | Nicotinic acid (niacin) | Charite University, Berlin, Germany | marketed | Lipid-modifying agent; B vitamin | GPR109A (HM74A receptor) | |
| Statin plus niacin ER/laropiprant | Statin plus niacin ER/laropiprant | University of Ioannina | marketed | Statin combined with niacin ER and DP1 antagonist | HMG-CoA reductase (statin component); GPR109A/PUMA-G (niacin component); DP1 receptor (laropiprant component) | |
| Niacin Extended Release/Lovastatin | Niacin Extended Release/Lovastatin | In His Image | marketed | Statin/Niacin combination; Lipid-modifying agent | HMG-CoA reductase (lovastatin); GPR109A/PUMA-G receptor (niacin) | |
| Niacin plus laropiprant | Niacin plus laropiprant | Institut Investigacio Sanitaria Pere Virgili | marketed | Lipid-modifying agent combination | DP1 receptor (laropiprant component); niacin acts on GPR109A and other pathways | |
| Slo-Niacin, atorvastatin | Slo-Niacin, atorvastatin | University of Washington | marketed | Niacin derivative and HMG-CoA reductase inhibitor (statin combination) | Nicotinic acid receptor (GPR109A) and HMG-CoA reductase | |
| nicotinic acid/laropiprant | nicotinic acid/laropiprant | Manchester University NHS Foundation Trust | marketed | Lipid-modifying agent / Antilipemic | GPR109A receptor (laropiprant component); nicotinic acid acts on multiple lipid metabolism pathways |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (lipid-regulating agent class)
- GWT-TUD GmbH · 1 drug in this class
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Cite this brief
Drug Landscape (2026). nicotine acid — Competitive Intelligence Brief. https://druglandscape.com/ci/nicotine-acid. Accessed 2026-05-14.
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