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nicotine acid — Competitive Intelligence Brief

nicotine acid (nicotine acid) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: lipid-regulating agent. Area: Cardiovascular.

phase 3 lipid-regulating agent GPR109A Cardiovascular Small molecule Live · refreshed every 30 min

Target snapshot

nicotine acid (nicotine acid) — GWT-TUD GmbH. Nicotine acid, also known as niacin, primarily functions by reducing the production of very-low-density lipoprotein (VLDL) and low-density lipoprotein (LDL) cholesterol in the liver.

Comparator set (6 drugs)

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DrugGenericSponsorPhaseClassTargetApproval / PDUFA
nicotine acid TARGET nicotine acid GWT-TUD GmbH phase 3 lipid-regulating agent GPR109A
Nicotinic acid (niacin) Nicotinic acid (niacin) Charite University, Berlin, Germany marketed Lipid-modifying agent; B vitamin GPR109A (HM74A receptor)
Statin plus niacin ER/laropiprant Statin plus niacin ER/laropiprant University of Ioannina marketed Statin combined with niacin ER and DP1 antagonist HMG-CoA reductase (statin component); GPR109A/PUMA-G (niacin component); DP1 receptor (laropiprant component)
Niacin Extended Release/Lovastatin Niacin Extended Release/Lovastatin In His Image marketed Statin/Niacin combination; Lipid-modifying agent HMG-CoA reductase (lovastatin); GPR109A/PUMA-G receptor (niacin)
Niacin plus laropiprant Niacin plus laropiprant Institut Investigacio Sanitaria Pere Virgili marketed Lipid-modifying agent combination DP1 receptor (laropiprant component); niacin acts on GPR109A and other pathways
Slo-Niacin, atorvastatin Slo-Niacin, atorvastatin University of Washington marketed Niacin derivative and HMG-CoA reductase inhibitor (statin combination) Nicotinic acid receptor (GPR109A) and HMG-CoA reductase
nicotinic acid/laropiprant nicotinic acid/laropiprant Manchester University NHS Foundation Trust marketed Lipid-modifying agent / Antilipemic GPR109A receptor (laropiprant component); nicotinic acid acts on multiple lipid metabolism pathways

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (lipid-regulating agent class)

  1. GWT-TUD GmbH · 1 drug in this class

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Cite this brief

Drug Landscape (2026). nicotine acid — Competitive Intelligence Brief. https://druglandscape.com/ci/nicotine-acid. Accessed 2026-05-14.

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