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Myrbetriq — Competitive Intelligence Brief
marketed
beta3-Adrenergic Agonist [EPC]
Beta-3 adrenergic receptor
Urology
Small molecule
Live · refreshed every 30 min
Target snapshot
Myrbetriq (MIRABEGRON) — Apgdi. Myrbetriq works by activating the beta-3 adrenergic receptor in the bladder muscle, leading to relaxation and improved bladder control.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Myrbetriq TARGET | MIRABEGRON | Apgdi | marketed | beta3-Adrenergic Agonist [EPC] | Beta-3 adrenergic receptor | 2012-01-01 |
| tolterodine , mirabegron | tolterodine , mirabegron | Far Eastern Memorial Hospital | marketed | Antimuscarinic and beta-3 adrenergic agonist combination | Muscarinic M3 receptor and beta-3 adrenergic receptor | |
| Solifenacin + Mirabegron | Solifenacin + Mirabegron | University of Aarhus | marketed | Antimuscarinic + Beta-3 adrenergic agonist combination | M3 muscarinic receptor (solifenacin) and beta-3 adrenergic receptor (mirabegron) | |
| daytime dosing of mirabegron | daytime dosing of mirabegron | Far Eastern Memorial Hospital | marketed | Beta-3 adrenergic receptor agonist | Beta-3 adrenergic receptor (ADRB3) | |
| nighttime dosing of mirabegron | nighttime dosing of mirabegron | Far Eastern Memorial Hospital | marketed | Beta-3 adrenergic receptor agonist | Beta-3 adrenergic receptor (ADRB3) | |
| Brovana | Brovana | Wake Forest University Health Sciences | marketed | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Beta-3 adrenergic receptor | ||
| Mirabegron tablet | Mirabegron tablet | Astellas Pharma Inc | marketed | Beta-3 adrenergic receptor agonist | Beta-3 adrenergic receptor (ADRB3) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (beta3-Adrenergic Agonist [EPC] class)
- · 1 drug in this class
- Apgdi · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Myrbetriq — Competitive Intelligence Brief. https://druglandscape.com/ci/mirabegron. Accessed 2026-05-13.
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