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Mineralocorticoid receptor antagonist potassium-canrenoate — Competitive Intelligence Brief
phase 3
Mineralocorticoid receptor antagonist
Mineralocorticoid receptor (MR)
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Mineralocorticoid receptor antagonist potassium-canrenoate (Mineralocorticoid receptor antagonist potassium-canrenoate) — University College, London. Potassium-canrenoate blocks mineralocorticoid receptors to reduce sodium reabsorption and potassium excretion in the kidney, lowering blood pressure and reducing fluid retention.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Mineralocorticoid receptor antagonist potassium-canrenoate TARGET | Mineralocorticoid receptor antagonist potassium-canrenoate | University College, London | phase 3 | Mineralocorticoid receptor antagonist | Mineralocorticoid receptor (MR) | |
| Eplerenone (Night-time) | Eplerenone (Night-time) | Vanderbilt University Medical Center | marketed | Selective aldosterone antagonist (mineralocorticoid receptor antagonist) | Mineralocorticoid receptor (MR) | |
| Ambrisentan plus Spironolactone | Ambrisentan plus Spironolactone | Brigham and Women's Hospital | marketed | Endothelin receptor antagonist + Mineralocorticoid receptor antagonist combination | Endothelin-1 receptor (ETA/ETB) + Mineralocorticoid receptor | |
| Mineralocorticoid Receptor Antagonist | Mineralocorticoid Receptor Antagonist | Cheng-Hsin General Hospital | marketed | Mineralocorticoid receptor antagonist | Mineralocorticoid receptor (MR) | |
| Finerenone (BAY 94-8862) | Finerenone (BAY 94-8862) | University Medical Center Groningen | marketed | Non-steroidal mineralocorticoid receptor antagonist | Mineralocorticoid receptor (MR) | |
| Propranolol - Spironolactone | Propranolol - Spironolactone | University Hospital, Angers | marketed | Beta-blocker and mineralocorticoid receptor antagonist combination | Beta-adrenergic receptors (propranolol); mineralocorticoid receptor (spironolactone) | |
| ACEI / ARB+finerenone | ACEI / ARB+finerenone | Capital Institute of Pediatrics, China | marketed | ACE inhibitor / ARB + non-steroidal mineralocorticoid receptor antagonist combination | Angiotensin-converting enzyme / Angiotensin II type 1 receptor + Mineralocorticoid receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Mineralocorticoid receptor antagonist class)
- Bayer · 1 drug in this class
- Cheng-Hsin General Hospital · 1 drug in this class
- Daiichi Sankyo Co., Ltd. · 1 drug in this class
- Kowa Company, Ltd. · 1 drug in this class
- University College, London · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Mineralocorticoid receptor antagonist potassium-canrenoate — Competitive Intelligence Brief. https://druglandscape.com/ci/mineralocorticoid-receptor-antagonist-potassium-canrenoate. Accessed 2026-05-17.
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