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mercaptopurine tablet — Competitive Intelligence Brief
phase 3
Purine analog antimetabolite
Hypoxanthine-guanine phosphoribosyltransferase (HGPRT), thiopurine methyltransferase (TPMT), and purine synthesis pathway enzymes
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
mercaptopurine tablet (mercaptopurine tablet) — National Cancer Institute (NCI). Mercaptopurine is a purine analog that inhibits nucleotide synthesis and DNA replication, leading to cell death in rapidly dividing cells.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| mercaptopurine tablet TARGET | mercaptopurine tablet | National Cancer Institute (NCI) | phase 3 | Purine analog antimetabolite | Hypoxanthine-guanine phosphoribosyltransferase (HGPRT), thiopurine methyltransferase (TPMT), and purine synthesis pathway enzymes | |
| Fludarabine (Flud) | Fludarabine (Flud) | Technische Universität Dresden | marketed | Purine analog antimetabolite | Ribonucleotide reductase, DNA polymerase | |
| 6MP | 6MP | South China Children's Leukemia Group | marketed | Purine analog antimetabolite | Hypoxanthine-guanine phosphoribosyltransferase (HGPRT), inosine monophosphate dehydrogenase (IMPDH) | |
| Fludarabine (Bayer) | Fludarabine (Bayer) | Chinese PLA General Hospital | marketed | Purine analog antimetabolite | Ribonucleotide reductase, DNA polymerase | |
| Mercaptopurine, Imatinib | Mercaptopurine, Imatinib | St. Jude Children's Research Hospital | phase 3 | Purine analog antimetabolite and tyrosine kinase inhibitor combination | Purine metabolism enzymes (mercaptopurine); BCR-ABL, c-KIT, PDGFR (imatinib) | |
| Fludarabine mono | Fludarabine mono | German CLL Study Group | phase 3 | Purine analog antimetabolite | Ribonucleotide reductase; DNA polymerase | |
| Experimental (fludarabine) | Experimental (fludarabine) | French Innovative Leukemia Organisation | phase 3 | Purine analog antimetabolite | Ribonucleotide reductase, DNA polymerase |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Purine analog antimetabolite class)
- Academisch Medisch Centrum - Universiteit van Amsterdam (AMC-UvA) · 1 drug in this class
- Chia Tai Tianqing Pharmaceutical Group Co., Ltd. · 1 drug in this class
- Chinese PLA General Hospital · 1 drug in this class
- French Innovative Leukemia Organisation · 1 drug in this class
- German CLL Study Group · 1 drug in this class
- National Cancer Institute (NCI) · 1 drug in this class
- South China Children's Leukemia Group · 1 drug in this class
- Technische Universität Dresden · 1 drug in this class
- University of California, San Francisco · 1 drug in this class
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Cite this brief
Drug Landscape (2026). mercaptopurine tablet — Competitive Intelligence Brief. https://druglandscape.com/ci/mercaptopurine-tablet. Accessed 2026-05-17.
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