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Mercaptopurine, Imatinib — Competitive Intelligence Brief

Mercaptopurine, Imatinib (Mercaptopurine, Imatinib) competitive landscape: 0 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Purine analog antimetabolite and tyrosine kinase inhibitor combination. Area: Oncology.

phase 3 Purine analog antimetabolite and tyrosine kinase inhibitor combination Purine metabolism enzymes (mercaptopurine); BCR-ABL, c-KIT, PDGFR (imatinib) Oncology Small molecule Live · refreshed every 30 min

Target snapshot

Mercaptopurine, Imatinib (Mercaptopurine, Imatinib) — St. Jude Children's Research Hospital. Mercaptopurine and imatinib work together as a combination therapy: mercaptopurine is a purine analog that inhibits nucleotide synthesis to kill rapidly dividing cells, while imatinib is a tyrosine kinase inhibitor that blocks BCR-ABL and other oncogenic kinases.

Comparator set

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Mercaptopurine, Imatinib TARGET Mercaptopurine, Imatinib St. Jude Children's Research Hospital phase 3 Purine analog antimetabolite and tyrosine kinase inhibitor combination Purine metabolism enzymes (mercaptopurine); BCR-ABL, c-KIT, PDGFR (imatinib)

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Purine analog antimetabolite and tyrosine kinase inhibitor combination class)

  1. St. Jude Children's Research Hospital · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Mercaptopurine, Imatinib — Competitive Intelligence Brief. https://druglandscape.com/ci/mercaptopurine-imatinib. Accessed 2026-05-17.

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